SCHEMBL5599763

SCHEMBL5599763

O=C(C[C@H]1N(C(=O)c2cccc(F)c2F)c2ccc(Cl)cc2C12CCNCC2)c1ccc(Cl)cc1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 3/20 0.38
PTGDR2 Q9Y5Y4 4/20 0.35
GNRHR P30968 1/20 0.34
KCNH2 Q12809 1/20 0.34
MGLL Q99685 2/20 0.33
P2RX7 Q99572 1/20 0.33
CHRM1 P11229 4/20 0.33
CHRM3 P20309 3/20 0.33
ALDH1A1 P00352 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
HPGD P15428 1/20 0.32
CHRM2 P08172 1/20 0.32
CHRM4 P08173 1/20 0.32
CHRM5 P08912 1/20 0.32
MCHR1 Q99705 1/20 0.32
AVPR2 P30518 1/20 0.32
AVPR1A P37288 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5599571 0.96 PTGDR2 (0.37) DRD2PTGDR2GNRHRKCNH2P2RX7
SCHEMBL5780226 0.93 CDYL (0.35) DRD2PTGDR2GNRHRKCNH2ALDH1A1
SCHEMBL5599828 0.90 CHRM1 (0.38) DRD2GNRHRKCNH2MGLLCHRM1
SCHEMBL5599289 0.85 DRD2 (0.37) DRD2PTGDR2GNRHRKCNH2P2RX7
SCHEMBL5600563 0.85 TSHR (0.36) DRD2PTGDR2P2RX7CHRM1CHRM3
SCHEMBL5780173 0.84 DRD2 (0.36) DRD2PTGDR2GNRHRKCNH2P2RX7
SCHEMBL5783150 0.82 PTGDR2 (0.36) DRD2PTGDR2P2RX7CHRM1CHRM3
SCHEMBL5779582 0.82 P2RX7 (0.41) DRD2PTGDR2GNRHRKCNH2P2RX7
SCHEMBL5782575 0.82 GPR183 (0.34) DRD2PTGDR2P2RX7CHRM1CHRM3
SCHEMBL5599553 0.81 PTGDR2 (0.33) DRD2PTGDR2GNRHRKCNH2P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005063745-A9 NOVEL SPIROINDOLINE OR SPIROISOQUINOLINE COMPOUNDS, METHODS OF USE AND COMPOSITIONS THEREOF ARENA PHARM INC (US) 2007-02-01 WO claimed