SCHEMBL5600154

SCHEMBL5600154

CCCCn1ccnc1Cc1ccc(Cl)c(Cl)c1O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.48
POLB P06746 1/20 0.48
KMT2A Q03164 1/20 0.48
TLR8 Q9NR97 2/20 0.39
KCNH2 Q12809 6/20 0.38
DRD2 P14416 1/20 0.34
DRD3 P35462 1/20 0.34
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA3 P07451 1/20 0.34
CA4 P22748 1/20 0.34
CA6 P23280 1/20 0.34
CA5A P35218 1/20 0.34
CA7 P43166 1/20 0.34
CA9 Q16790 1/20 0.34
CA13 Q8N1Q1 1/20 0.34
CA14 Q9ULX7 1/20 0.34
CA5B Q9Y2D0 1/20 0.34
AGTR1 P30556 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6649403 0.82 KMT2A (0.39) ALDH1A1KMT2ACA12CA1CA2
SCHEMBL6651569 0.81 KMT2A (0.47) ALDH1A1POLBKMT2ATLR8KCNH2
SCHEMBL9269515 0.80 KMT2A (0.51) ALDH1A1POLBKMT2ATLR8DRD2
SCHEMBL6115119 0.78 ALDH1A1 (0.69) ALDH1A1POLBKMT2ATLR8KCNH2
SCHEMBL6648269 0.77 KMT2A (0.46) ALDH1A1POLBKMT2ATLR8KCNH2
SCHEMBL6651433 0.73 KMT2A (0.43) ALDH1A1POLBKMT2ATLR8
SCHEMBL5655366 0.72 ALDH1A1 (0.59) ALDH1A1POLBKMT2ATLR8KCNH2
SCHEMBL28748507 0.72 ALDH1A1 (0.56) ALDH1A1POLBKMT2ATLR8AGTR1
SCHEMBL329466 0.71 ALDH1A1 (0.63) ALDH1A1POLBKMT2ATLR8KCNH2
SCHEMBL9935809 0.71 ALDH1A1 (0.63) ALDH1A1POLBKMT2ATLR8KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1103243-B1 UTILIZATION OF ARYL(OR HETEROARYL)AZOLYLCARBINOL DERIVATIVES FOR THE TREATMENT OF TROUBLES MEDIATED BY AN EXCESS OF SUBSTANCE P ESTEVE LABOR DR (ES) 2004-01-07 EP claimed
EP-1746986-A1 ACTIVE SUBSTANCE COMBINATION COMPRISING A CARBINOL COMBINED TO AT LEAST AN NSAID LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2007-01-31 EP disclosed
WO-2005097099-A1 ACTIVE SUBSTANCE COMBINATION COMPRISING A CARBINOL COMBINED TO AT LEAST AN NSAID LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2005-10-20 WO disclosed