SCHEMBL5607313

SCHEMBL5607313

CCCCn1sc(-c2ccccc2)c(Nc2ccc3oc(C(C)=O)cc3c2)c1=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.38
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 2/20 0.38
HPGD P15428 2/20 0.38
LMNA P02545 1/20 0.38
GLA P06280 1/20 0.38
GAA P10253 1/20 0.38
CASP1 P29466 1/20 0.38
BRCA1 P38398 1/20 0.38
CASP7 P55210 1/20 0.38
HSD17B10 Q99714 1/20 0.38
NPC1 O15118 5/20 0.37
RAB9A P51151 5/20 0.37
MAPK1 P28482 1/20 0.37
P2RX3 P56373 5/20 0.35
HDAC3 O15379 1/20 0.35
IKBKB O14920 1/20 0.34
SYK P43405 2/20 0.33
L3MBTL1 Q9Y468 3/20 0.33
MEN1 O00255 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5606136 0.86 SMN1; SMN2 (0.43) SMN1; SMN2KDM4EALDH1A1HPGDLMNA
SCHEMBL5606238 0.78 PGR (0.38) ALDH1A1HPGDNPC1RAB9AP2RX3
SCHEMBL5657430 0.77 EPHX1 (0.40) NPC1RAB9AP2RX3MAPT
SCHEMBL3487918 0.76 SMN1; SMN2 (0.38) SMN1; SMN2KDM4EALDH1A1HPGDLMNA
SCHEMBL5613996 0.72 MAPT (0.46) SMN1; SMN2KDM4EALDH1A1LMNAGAA
SCHEMBL5613761 0.72 PSMB8 (0.41) SMN1; SMN2KDM4EALDH1A1HPGDLMNA
SCHEMBL5613942 0.71 BPTF (0.43)
SCHEMBL5606522 0.71 PLK1 (0.41) SMN1; SMN2ALDH1A1GAAHDAC3MEN1
SCHEMBL5607253 0.71 MAPT (0.38) ALDH1A1LMNAP2RX3MEN1KMT2A
SCHEMBL17844161 0.70 FAAH (0.44) SMN1; SMN2KDM4EALDH1A1HPGDLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1838686-A1 DERIVATIVES OF ISOTHIAZOL-3(2H)-ONE 1,1-DIOXIDES AS LIVER X RECEPTOR MODULATORS AstraZeneca AB (SE) 2007-10-03 EP claimed
WO-2006073363-A1 DERIVATIVES OF ISOTHIAZOL-3(2H)-ONE 1,1-DIOXIDES AS LIVER X RECEPTOR MODULATORS ASTRAZENECA AB (SE) 2006-07-13 WO claimed