SCHEMBL5608722

SCHEMBL5608722

O=CC(Br)c1cc(C(F)(F)F)ccc1F

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 3/20 0.43
TDO2 P48775 1/20 0.43
PDE2A O00408 4/20 0.40
MEN1 O00255 1/20 0.36
TSHR P16473 1/20 0.36
KMT2A Q03164 1/20 0.36
GSK3B P49841 1/20 0.36
GAA P10253 1/20 0.34
BACE1 P56817 1/20 0.33
ALOX5AP P20292 1/20 0.33
FEN1 P39748 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
MPL P40238 1/20 0.33
CES2 O00748 2/20 0.33
TMPRSS4 Q9NRS4 1/20 0.32
AHR P35869 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4963648 0.86 PDE2A (0.51) IDO1TDO2PDE2AGSK3BGAA
SCHEMBL20551557 0.86 PDE2A (0.51) IDO1TDO2PDE2AGSK3BGAA
SCHEMBL6446889 0.83 CES2 (0.43) IDO1TDO2PDE2AGSK3BCES2
SCHEMBL6448282 0.81 PDE2A (0.36) PDE2AMEN1KMT2AGSK3BCES2
SCHEMBL3248499 0.81 PDE2A (0.42) PDE2AMEN1TSHRKMT2AGSK3B
SCHEMBL27551257 0.79 PDE2A (0.47) IDO1TDO2PDE2AMEN1TSHR
SCHEMBL27490326 0.79 IDO1 (0.40) IDO1TDO2PDE2AMEN1TSHR
SCHEMBL6442608 0.78 CES2 (0.43) CES2
SCHEMBL20551270 0.78 CES2 (0.43) CES2
SCHEMBL17604466 0.77 DGAT1 (0.35) KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1749002-A1 PYRROLE OR IMIDAZOLE AMIDES FOR TREATING OBESITY F.HOFFMANN-LA ROCHE AG (CH) 2007-02-07 EP disclosed
WO-2005108393-A1 PYRROLE OR IMIDAZOLE AMIDES FOR TREATING OBESITY F. HOFFMANN-LA ROCHE AG (CH) 2005-11-17 WO disclosed