SCHEMBL6448282

SCHEMBL6448282

Cc1ccc(C(F)(F)F)cc1C(Br)C=O

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 4/20 0.36
NOTUM Q6P988 1/20 0.35
GSK3B P49841 1/20 0.35
TAS2R14 Q9NYV8 1/20 0.35
MAPT P10636 1/20 0.33
KIF11 P52732 1/20 0.33
KDM4E B2RXH2 1/20 0.32
MCL1 Q07820 1/20 0.32
MTOR P42345 1/20 0.32
CYP1A1 P04798 1/20 0.32
CYP1B1 Q16678 1/20 0.32
DAO P14920 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
NFE2L2 Q16236 1/20 0.32
CYP1A2 P05177 1/20 0.32
CES2 O00748 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27624247 0.85 PDE2A (0.40) PDE2ANOTUMTAS2R14MAPTKIF11
SCHEMBL6446889 0.81 CES2 (0.43) PDE2AGSK3BMAPTKIF11KDM4E
SCHEMBL5608722 0.81 IDO1 (0.43) PDE2AGSK3BMEN1KMT2ACES2
SCHEMBL3248499 0.80 PDE2A (0.42) PDE2AGSK3BMCL1MEN1KMT2A
SCHEMBL27624269 0.80 PDE2A (0.35) PDE2ANOTUMGSK3BTAS2R14MAPT
SCHEMBL4963648 0.78 PDE2A (0.51) PDE2AGSK3B
SCHEMBL20551557 0.78 PDE2A (0.51) PDE2AGSK3B
SCHEMBL6443794 0.77 HDAC4 (0.33) MAPTKDM4EMEN1KMT2ACES2
SCHEMBL929896 0.77 LMNA (0.38) MEN1KMT2ACYP1A2
SCHEMBL12306470 0.74 PDE2A (0.46) PDE2ANOTUMTAS2R14KIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1583742-A1 NOVEL CB 1 RECEPTOUR INVERSE AGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2005-10-12 EP disclosed
WO-2004060870-A1 NOVEL CB 1 RECEPTOUR INVERSE AGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2004-07-22 WO disclosed