SCHEMBL6446889

SCHEMBL6446889

O=CC(Br)c1cc(C(F)(F)F)ccc1C(F)(F)F

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.43
GSK3B P49841 1/20 0.36
PDE2A O00408 6/20 0.34
CYP26A1 O43174 1/20 0.33
CYP24A1 Q07973 1/20 0.33
KIF11 P52732 1/20 0.33
MAPT P10636 1/20 0.31
XBP1 P17861 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
IDO1 P14902 1/20 0.31
TDO2 P48775 1/20 0.31
PIM1 P11309 1/20 0.31
PIM2 Q9P1W9 1/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
HSD17B10 Q99714 1/20 0.31
PTPN5 P54829 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5608722 0.83 IDO1 (0.43) CES2GSK3BPDE2AIDO1TDO2
SCHEMBL6448282 0.81 PDE2A (0.36) CES2GSK3BPDE2AKIF11MAPT
SCHEMBL3248499 0.81 PDE2A (0.42) GSK3BPDE2AALDH1A1
SCHEMBL2954138 0.80 CES2 (0.46) CES2GSK3BPDE2AKIF11IDO1
SCHEMBL4963648 0.79 PDE2A (0.51) GSK3BPDE2AIDO1TDO2
SCHEMBL20551557 0.79 PDE2A (0.51) GSK3BPDE2AIDO1TDO2
SCHEMBL27643644 0.79 CES2 (0.40) CES2GSK3BPDE2ACYP26A1CYP24A1
SCHEMBL22717245 0.77 P2RX7 (0.47) CES2GSK3BPDE2AKIF11IDO1
SCHEMBL17698505 0.77 P2RX7 (0.47) CES2GSK3BPDE2AKIF11IDO1
SCHEMBL21495118 0.77 ACP3 (0.44) IDO1TDO2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1583742-A1 NOVEL CB 1 RECEPTOUR INVERSE AGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2005-10-12 EP disclosed
WO-2004060870-A1 NOVEL CB 1 RECEPTOUR INVERSE AGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2004-07-22 WO disclosed