SCHEMBL5609346

SCHEMBL5609346

CCc1cccc2ccn(-c3cc(C)cc(C)c3)c12

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.41
THRB P10828 1/20 0.41
COMT P21964 1/20 0.40
BACE1 P56817 1/20 0.35
RAPGEF4 Q8WZA2 1/20 0.34
TP53 P04637 1/20 0.34
IDH1 O75874 1/20 0.33
HCAR1 Q9BXC0 1/20 0.33
HPGD P15428 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
GABRA1 P14867 2/20 0.32
GABRB2 P47870 2/20 0.32
FFAR4 Q5NUL3 1/20 0.32
OXER1 Q8TDS5 1/20 0.32
DAO P14920 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1762891 0.72 MAPT (0.37) MAPTTHRBCOMTTP53HPGD
SCHEMBL11005480 0.71 CMA1 (0.48) BACE1GABRA1GABRB2OXER1
SCHEMBL5608903 0.70 PTK2 (0.54) MAPT
SCHEMBL6608085 0.69 GABRA1 (0.43) BACE1HPGDGABRA1GABRB2OXER1
SCHEMBL5216431 0.69 BIRC5 (0.55) MAPTCOMTRAPGEF4HPGDL3MBTL1
SCHEMBL15676807 0.69 BACE1 (0.48) BACE1HPGDGABRA1GABRB2OXER1
SCHEMBL11474556 0.67 ACHE (0.50) MAPTRAPGEF4TP53L3MBTL1GABRA1
SCHEMBL10296017 0.66 ROCK1 (0.50) MAPTTHRBCOMTHPGDL3MBTL1
SCHEMBL18617117 0.66 RAPGEF4 (0.55) RAPGEF4HPGDL3MBTL1
SCHEMBL27550174 0.66 OXER1 (0.51) BACE1L3MBTL1GABRA1GABRB2OXER1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1354887-B1 Ligands for metals and improved metal-catalyzed processes based thereon MASSACHUSETTS INST TECHNOLOGY (US) 2007-04-25 EP disclosed
EP-1097158-B1 LIGANDS FOR METALS AND METAL-CATALYZED PROCESSES MASSACHUSETTS INST TECHNOLOGY (US) 2006-01-25 EP disclosed
EP-1354887-A1 Ligands for metals and improved metal-catalyzed processes based thereon Massachusetts Insitute of Technology (US) 2003-10-22 EP disclosed
EP-1097158-A2 LIGANDS FOR METALS AND METAL-CATALYZED PROCESSES MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2001-05-09 EP disclosed
WO-2000002887-A2 LIGANDS FOR METALS AND METAL-CATALYZED PROCESSES MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2000-01-20 WO disclosed