SCHEMBL5611033

SCHEMBL5611033

Cc1c(NS(C)(=O)=O)[c]ccc1-c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 2/20 0.42
CKS1B P61024 1/20 0.39
GLO1 Q04760 1/20 0.39
SKP2 Q13309 1/20 0.39
PTGS2 P35354 4/20 0.39
ALOX5 P09917 1/20 0.39
CYP17A1 P05093 1/20 0.39
LMNA P02545 4/20 0.38
ALDH1A1 P00352 3/20 0.38
HSP90AA1 P07900 2/20 0.38
KDM4E B2RXH2 1/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
MCOLN3 Q8TDD5 3/20 0.37
GAA P10253 1/20 0.37
THRB P10828 1/20 0.37
CA12 O43570 1/20 0.37
CA2 P00918 1/20 0.37
CA9 Q16790 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21408573 0.81 KEAP1 (0.44) KEAP1CKS1BGLO1SKP2PTGS2
SCHEMBL16759968 0.72 KEAP1 (0.61) KEAP1CKS1BGLO1SKP2LMNA
SCHEMBL29788215 0.72 KEAP1 (0.61) KEAP1CKS1BGLO1SKP2LMNA
SCHEMBL11269403 0.70 PDCD1 (0.42) PTGS2LMNAALDH1A1KDM4EHPGD
SCHEMBL21408485 0.70 CKS1B (0.46) KEAP1CKS1BGLO1SKP2PTGS2
SCHEMBL28903467 0.68 KEAP1 (0.44) KEAP1LMNAKDM4EMAPTHPGD
SCHEMBL4533547 0.67 KDM1A (0.60) KEAP1CKS1BGLO1SKP2PTGS2
SCHEMBL31645593 0.67 KDM1A (0.60) KEAP1CKS1BGLO1SKP2PTGS2
SCHEMBL5611087 0.67 KEAP1 (0.43) KEAP1CKS1BGLO1SKP2PTGS2
SCHEMBL157836 0.66 KEAP1 (0.47) KEAP1GLO1PTGS2ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1861365-A1 N-SULPHONYLPYRROLES AND THEIR USE AS HISTONE DEACETYLASE INHIBITORS Nycomed GmbH (DE) 2007-12-05 EP disclosed
WO-2006097474-A1 N-SULPHONYLPYRROLES AND THEIR USE AS HISTONE DEACETYLASE INHIBITORS NYCOMED GMBH (DE) 2006-09-21 WO disclosed