SCHEMBL5611087

SCHEMBL5611087

Cc1[c]c(NS(C)(=O)=O)ccc1-c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.43
CKS1B P61024 1/20 0.43
GLO1 Q04760 1/20 0.43
SKP2 Q13309 1/20 0.43
CYP17A1 P05093 1/20 0.42
LMNA P02545 4/20 0.39
MCOLN3 Q8TDD5 3/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ALDH1A1 P00352 3/20 0.39
PTGS2 P35354 3/20 0.39
HSP90AA1 P07900 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
CA12 O43570 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
GAA P10253 1/20 0.38
THRB P10828 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3145873 0.74 NAPRT (0.43) LMNASMN1; SMN2ALDH1A1HSP90AA1KDM4E
SCHEMBL28430442 0.70 KEAP1 (0.46) KEAP1PTGS2GSK3AGSK3BNR3C2
SCHEMBL456233 0.70 ESR2 (0.38) ALDH1A1PTGS2HPGDALOX5L3MBTL1
SCHEMBL4371389 0.69 ESR2 (0.41) LMNAMCOLN3SMN1; SMN2ALDH1A1PTGS2
SCHEMBL4533547 0.68 KDM1A (0.60) KEAP1CKS1BGLO1SKP2LMNA
SCHEMBL31645593 0.68 KDM1A (0.60) KEAP1CKS1BGLO1SKP2LMNA
SCHEMBL5961725 0.68 KEAP1 (0.43) KEAP1GLO1NR3C2PGRNR3C1
Lithium SCHEMBL31041204 0.67 AURKA (0.59) KEAP1CYP17A1LMNAALDH1A1PTGS2
SCHEMBL16759968 0.67 KEAP1 (0.61) KEAP1CKS1BGLO1SKP2LMNA
SCHEMBL29788215 0.67 KEAP1 (0.61) KEAP1CKS1BGLO1SKP2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1861365-A1 N-SULPHONYLPYRROLES AND THEIR USE AS HISTONE DEACETYLASE INHIBITORS Nycomed GmbH (DE) 2007-12-05 EP disclosed
WO-2006097474-A1 N-SULPHONYLPYRROLES AND THEIR USE AS HISTONE DEACETYLASE INHIBITORS NYCOMED GMBH (DE) 2006-09-21 WO disclosed