SCHEMBL5611086

SCHEMBL5611086

CS(=O)(=O)NCc1[c]cccc1-c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.40
GRIA4 P48058 1/20 0.38
POLB P06746 2/20 0.38
KDM4E B2RXH2 1/20 0.38
TSHR P16473 1/20 0.38
RECQL P46063 1/20 0.38
BRD4 O60885 2/20 0.37
KMT2A Q03164 1/20 0.36
PDCD1 Q15116 2/20 0.35
CD274 Q9NZQ7 2/20 0.35
SETDB1 Q15047 1/20 0.35
HPGD P15428 2/20 0.33
CA12 O43570 1/20 0.33
CA2 P00918 1/20 0.33
LMNA P02545 1/20 0.33
CA9 Q16790 1/20 0.33
MCOLN3 Q8TDD5 1/20 0.33
CREBBP Q92793 1/20 0.33
KEAP1 Q14145 1/20 0.33
CKS1B P61024 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19692916 0.79 KDM4E (0.39) KDM4EKMT2APDCD1CD274HPGD
SCHEMBL3145870 0.76 MTNR1A (0.45) KDM4EKMT2APDCD1CD274HPGD
SCHEMBL12462407 0.76 SETDB1 (0.49) PTGS2GRIA4POLBKDM4ETSHR
SCHEMBL19693021 0.75 HRH1 (0.43) KDM4EPDCD1CD274LMNA
SCHEMBL1774729 0.73 DPP4 (0.36) PTGS2KMT2APDCD1CD274HPGD
SCHEMBL21408573 0.73 KEAP1 (0.44) PTGS2KDM4EHPGDCA12CA2
SCHEMBL5611030 0.72 SETDB1 (0.40) PTGS2GRIA4POLBKDM4ETSHR
SCHEMBL5796914 0.71 ALDH1A1 (0.41) TSHRKMT2APDCD1CD274HPGD
SCHEMBL21408620 0.71 MEN1 (0.49) KMT2APDCD1CD274LMNA
SCHEMBL457404 0.70 SMN1; SMN2 (0.36) PTGS2KDM4EPDCD1CD274HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1861365-A1 N-SULPHONYLPYRROLES AND THEIR USE AS HISTONE DEACETYLASE INHIBITORS Nycomed GmbH (DE) 2007-12-05 EP disclosed
WO-2006097474-A1 N-SULPHONYLPYRROLES AND THEIR USE AS HISTONE DEACETYLASE INHIBITORS NYCOMED GMBH (DE) 2006-09-21 WO disclosed