SCHEMBL5614482

SCHEMBL5614482

CC(C)(C)OC(=O)C(N)=Cc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.45
MEN1 O00255 1/20 0.45
AKR1C3 P42330 1/20 0.43
MCL1 Q07820 1/20 0.41
CYP2C19 P33261 1/20 0.41
TSHR P16473 3/20 0.41
NPC1 O15118 1/20 0.41
ALDH1A1 P00352 2/20 0.39
MAPT P10636 1/20 0.39
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
AKR1C1 Q04828 1/20 0.38
RECQL P46063 1/20 0.38
HTT P42858 1/20 0.37
EGFR P00533 1/20 0.37
FBP1 P09467 2/20 0.36
HSD17B10 Q99714 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
NR1I2 O75469 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13241270 0.84 MEN1 (0.58) KMT2AMEN1AKR1C3CYP2C19TSHR
SCHEMBL1905155 0.82 MEN1 (0.47) KMT2AMEN1AKR1C3CYP2C19TSHR
SCHEMBL20853874 0.81 AKR1C3 (0.58) KMT2AMEN1AKR1C3TSHRNPC1
SCHEMBL28915528 0.81 AKR1C3 (0.58) KMT2AMEN1AKR1C3TSHRNPC1
Dehydrophenylalanine Methyl Ester SCHEMBL6947584 0.80 MEN1 (0.49) KMT2AMEN1AKR1C3MCL1TSHR
Dehydrophenylalanine Methyl Ester SCHEMBL6947585 0.80 MEN1 (0.49) KMT2AMEN1AKR1C3MCL1TSHR
SCHEMBL26080824 0.79 MEN1 (0.53) KMT2AMEN1AKR1C3CYP2C19TSHR
Dehydrophenylalanine Methyl Ester SCHEMBL27965511 0.79 MEN1 (0.47) KMT2AMEN1AKR1C3MCL1TSHR
SCHEMBL3227832 0.78 MEN1 (0.51) KMT2AMEN1AKR1C3MAPTHTT
SCHEMBL2409609 0.78 ABCG2 (0.47) KMT2AMEN1AKR1C3TSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108794474-B Evodiamine derivative with multi-target antitumor activity and preparation method and application thereof 中国人民解放军第二军医大学 2022-03-18 CN claimed
CN-108794474-A Rutaecarpin derivative and its preparation method and application with multiple target point antitumor activity 中国人民解放军第二军医大学 2018-11-13 CN claimed
CN-108794474-A Rutaecarpin derivative and its preparation method and application with multiple target point antitumor activity 中国人民解放军第二军医大学 2018-11-13 CN disclosed
US-7229574-B2 Method of making novel water-soluble and self-doped polyaniline graft copolymers SEOUL NATIONAL UNIVERSITY INDUSTRY FOUNDATION (KR) 2007-06-12 US disclosed
US-20060175580-A1 Novel water-soluble and self-doped polyaniline graft copolymers SEOUL NATIONAL UNIVERSITY INDUSTRY FOUNDATION (KR) 2006-08-10 US disclosed
WO-2005068551-A1 A EXFOLIATED NANO-COMPOSITE FROM POLYANILINE GRAFT COPOLYMER/CLAY SEOUL NATIONAL UNIVERSITY INDUSTRY FOUNDATION (KR) 2005-07-28 WO disclosed