SCHEMBL5615330

SCHEMBL5615330

CC(C)[C@H](N)C(=O)ON1C(=O)CCC1=O

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SLC7A5 Q01650 1/20 0.35
MGLL Q99685 2/20 0.33
DPP4 P27487 1/20 0.30
HTR1A P08908 1/20 0.30
TBXA2R P21731 1/20 0.30
PTGS1 P23219 1/20 0.30
OPRM1 P35372 1/20 0.30
KCNH2 Q12809 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24576662 1.00 SLC7A5 (0.35) SLC7A5MGLLDPP4HTR1ATBXA2R
SCHEMBL8478185 1.00 SLC7A5 (0.35) SLC7A5MGLLDPP4HTR1ATBXA2R
SCHEMBL13061953 0.85 MGLL (0.34) MGLLDPP4
SCHEMBL356572 0.85 MGLL (0.34) MGLLDPP4
SCHEMBL10869514 0.85 MGLL (0.34) MGLLDPP4
SCHEMBL14804761 0.83 DPP4 (0.41) DPP4
SCHEMBL7397688 0.83 DPP4 (0.41) DPP4
SCHEMBL22954473 0.81 MGLL (0.34) MGLL
SCHEMBL13463250 0.81 MGLL (0.34) MGLL
SCHEMBL12092206 0.81 MGLL (0.34) MGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 50 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260091024-A1 PRODRUGS OF RILUZOLE AND THEIR METHOD OF USE BIOHAVEN THERAPEUTICS LTD (US) 2026-04-02 US disclosed
US-20260041673-A1 PRODRUGS OF RILUZOLE AND THEIR METHOD OF USE BIOHAVEN THERAPEUTICS LTD (US) 2026-02-12 US disclosed
US-12472165-B2 Riluzole prodrugs and their use BIOHAVEN THERAPEUTICS LTD. (VG) 2025-11-18 US disclosed
US-20250332148-A1 RILUZOLE PRODRUGS AND THEIR USE BIOHAVEN THERAPEUTICS LTD (US) 2025-10-30 US disclosed
US-12295942-B2 Riluzole prodrugs and their use BIOHAVEN THERAPEUTICS LTD. (VG) 2025-05-13 US disclosed
US-12213965-B2 Riluzole prodrugs and their use BIOHAVEN THERAPEUTICS LTD. (VG) 2025-02-04 US disclosed
CN-118846112-A Cysteine engineered antibody-toxin conjugates and methods of making same 四川百利药业有限责任公司 2024-10-29 CN disclosed
US-12005046-B2 Riluzole prodrugs and their use BIOHAVEN THERAPEUTICS LTD. (US) 2024-06-11 US disclosed
US-12005047-B2 Riluzole prodrugs and their use BIOHAVEN THERAPEUTICS LTD. (US) 2024-06-11 US disclosed
US-20240091205-A1 PRODRUGS OF RILUZOLE AND THEIR METHOD OF USE BEETLEJUICE SA LLC, AS PURCHASER AGENT 2024-03-21 US disclosed
US-20150132324-A1 TUBULYSIN COMPOUNDS, METHODS OF MAKING AND USE BRISTOL-MYERS SQUIBB COMPANY 2015-05-14 US disclosed
US-8980824-B2 Tubulysin compounds, methods of making and use BRISTOL-MYERS SQUIBB COMPANY (US) 2015-03-17 US disclosed
WO-2014126836-A1 TUBULYSIN COMPOUNDS, METHODS OF MAKING AND USE BRISTOL-MYERS SQUIBB COMPANY (US) 2014-08-21 WO disclosed
US-20140227295-A1 TUBULYSIN COMPOUNDS, METHODS OF MAKING AND USE BRISTOL-MYERS SQUIBB COMPANY 2014-08-14 US disclosed
US-20140227298-A1 TUBULYSIN COMPOUNDS, METHODS OF MAKING AND USE BRISTOL-MYERS SQUIBB COMPANY 2014-08-14 US disclosed
EP-1749007-A2 MACROCYCLIC COMPOUNDS AS INHIBITORS OF VIRAL REPLICATION Intermune, Inc. (US) 2007-02-07 EP disclosed
EP-1680137-A2 MACROCYCLIC CARBOXYLIC ACIDS AND ACYLSULFONAMIDES AS INHIBITORS OF HCV REPLICATION Intermune, Inc. (US) 2006-07-19 EP disclosed
WO-2005095403-A2 MACROCYCLIC COMPOUNDS AS INHIBITORS OF VIRAL REPLICATION INTERMUNE, INC. (US) 2005-10-13 WO disclosed
WO-2005037214-A2 MACROCYCLIC CARBOXYLIC ACIDS AND ACYLSULFONAMIDES AS INHIBITORS OF HCV REPLICATION INTERMUNE, INC. (US) 2005-04-28 WO disclosed
US-5955501-A DERIVED FROM PHORBOIDS OF THE DITERPENE- AND BENZOLACTAM-CLASSES. PROCYON PHARMACEUTICALS, INC. (US) 1999-09-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (12 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260091024-A1 PRODRUGS OF RILUZOLE AND THEIR METHOD OF USE IL6ST, GFRA3, GFRA1 SLC7A5 1202/4885MGLL 1184/4885DPP4 1982/4885
US-20150132324-A1 TUBULYSIN COMPOUNDS, METHODS OF MAKING AND USE CCNB1, CCNB3, CCNB2 SLC7A5 2274/4885MGLL 4835/4885DPP4 3888/4885
US-12005046-B2 Riluzole prodrugs and their use APEH, ALDH1A2, UGT1A9 SLC7A5 3261/4885MGLL 126/4885DPP4 225/4885
US-20140227298-A1 TUBULYSIN COMPOUNDS, METHODS OF MAKING AND USE CCNB3, CCNB1, CCNB2 SLC7A5 2237/4885MGLL 4844/4885DPP4 4179/4885
US-12005047-B2 Riluzole prodrugs and their use APEH, ALDH1A2, UGT1A9 SLC7A5 3261/4885MGLL 126/4885DPP4 225/4885
US-20260041673-A1 PRODRUGS OF RILUZOLE AND THEIR METHOD OF USE GFRA3, IL6ST, GFRA1 SLC7A5 877/4885MGLL 1124/4885DPP4 1899/4885
US-20140227295-A1 TUBULYSIN COMPOUNDS, METHODS OF MAKING AND USE CCNB1, CCNB3, CCNB2 SLC7A5 2274/4885MGLL 4835/4885DPP4 3888/4885
US-12472165-B2 Riluzole prodrugs and their use APEH, ALDH1A2, UGT1A9 SLC7A5 3261/4885MGLL 126/4885DPP4 225/4885
US-12295942-B2 Riluzole prodrugs and their use APEH, ALDH1A2, UGT1A9 SLC7A5 3261/4885MGLL 126/4885DPP4 225/4885
US-20240091205-A1 PRODRUGS OF RILUZOLE AND THEIR METHOD OF USE APEH, UGT1A9, ALDH3A1 SLC7A5 2829/4885MGLL 196/4885DPP4 326/4885
US-20250332148-A1 RILUZOLE PRODRUGS AND THEIR USE APEH, ALDH1A2, UGT1A9 SLC7A5 3261/4885MGLL 126/4885DPP4 225/4885
US-12213965-B2 Riluzole prodrugs and their use APEH, ALDH1A2, UGT1A9 SLC7A5 3261/4885MGLL 126/4885DPP4 225/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.