SCHEMBL5618229

SCHEMBL5618229

OC/C(=C/F)Cc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BTN3A1 O00481 2/20 0.47
CES1 P23141 2/20 0.43
CES2 O00748 1/20 0.43
AKR1B1 P15121 1/20 0.43
TSHR P16473 2/20 0.42
ALDH1A1 P00352 1/20 0.39
MAPK1 P28482 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
MAOB P27338 3/20 0.39
AOC2 O75106 2/20 0.39
MAOA P21397 2/20 0.39
DAO P14920 1/20 0.39
PAM P19021 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5618233 1.00 BTN3A1 (0.47) BTN3A1CES1CES2AKR1B1TSHR
SCHEMBL10727744 1.00 BTN3A1 (0.47) BTN3A1CES1CES2AKR1B1TSHR
SCHEMBL27912802 0.86 CES1 (0.46) CES1CES2AKR1B1TSHRALDH1A1
SCHEMBL10722411 0.81 AOC2 (0.55) CES1CES2AKR1B1ALDH1A1MAPK1
SCHEMBL10724983 0.81 AOC2 (0.55) CES1CES2AKR1B1ALDH1A1MAPK1
SCHEMBL10722397 0.81 AOC2 (0.55) CES1CES2AKR1B1ALDH1A1MAPK1
SCHEMBL13884200 0.81 CES1 (0.41) CES1CES2AKR1B1TSHRALDH1A1
Ammonia Solution, Strong SCHEMBL11133048 0.79 AOC2 (0.53) CES1CES2AKR1B1ALDH1A1MAPK1
SCHEMBL10723401 0.79 BTN3A1 (0.50) BTN3A1L3MBTL1TDP1MEN1KMT2A
SCHEMBL10723473 0.79 BTN3A1 (0.50) BTN3A1MAPK1L3MBTL1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070078172-A1 MAO-B INHIBITORS USEFUL FOR TREATING OBESITY JENRIN DISCOVERY (US) 2007-04-05 US claimed
WO-2006138475-A2 MAO-B INHIBITORS USEFUL FOR TREATING OBESITY JENRIN DISCOVERY (US) 2006-12-28 WO claimed
US-4454158-A Allyl amine MAO inhibitors MERRELL TORAUDE ET COMPAGNIE (FR) 1984-06-12 US claimed
US-20070078172-A1 MAO-B INHIBITORS USEFUL FOR TREATING OBESITY JENRIN DISCOVERY (US) 2007-04-05 US disclosed
WO-2006138475-A2 MAO-B INHIBITORS USEFUL FOR TREATING OBESITY JENRIN DISCOVERY (US) 2006-12-28 WO disclosed
EP-0067105-B1 ALLYL AMINE MAO INHIBITORS MERRELL DOW FRANCE ET CIE (FR) 1987-09-23 EP disclosed
US-4454158-A Allyl amine MAO inhibitors MERRELL TORAUDE ET COMPAGNIE (FR) 1984-06-12 US disclosed
EP-0067105-A2 Allyl amine MAO inhibitors MERRELL DOW FRANCE ET CIE (FR) 1982-12-15 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070078172-A1 MAO-B INHIBITORS USEFUL FOR TREATING OBESITY MAOB, MAOA, GPR119 BTN3A1 3679/4885CES1 86/4885CES2 53/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.