SCHEMBL5625798

SCHEMBL5625798

CCn1c(Cn2ccnc2-c2c[c]ccc2)nc2cc(F)ccc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 3/20 0.40
CYP11B1 P15538 2/20 0.40
RPS6KA5 O75582 1/20 0.37
AGTR1 P30556 1/20 0.36
AGTR2 P50052 1/20 0.36
MAP4K1 Q92918 2/20 0.35
NLRP3 Q96P20 1/20 0.35
ALDH1A1 P00352 3/20 0.35
GAA P10253 2/20 0.35
PKM P14618 1/20 0.35
CRHBP P24387 1/20 0.35
CRHR2 Q13324 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
RAB9A P51151 1/20 0.34
TBXA2R P21731 4/20 0.34
KDM4E B2RXH2 2/20 0.34
MAPT P10636 2/20 0.34
MAPK1 P28482 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
HSD17B10 Q99714 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3063221 0.88 NLRP3 (0.43) CYP11B2CYP11B1RPS6KA5AGTR1AGTR2
SCHEMBL3059869 0.83 CYP11B1 (0.41) CYP11B2CYP11B1RPS6KA5AGTR1AGTR2
SCHEMBL3050438 0.83 CYP11B1 (0.41) CYP11B2CYP11B1RPS6KA5AGTR1AGTR2
SCHEMBL3070468 0.83 MAPT (0.46) CYP11B2CYP11B1RPS6KA5AGTR1AGTR2
SCHEMBL3065899 0.83 CYP11B2 (0.39) CYP11B2CYP11B1RPS6KA5MAP4K1ALDH1A1
SCHEMBL3061263 0.83 CYP11B2 (0.42) CYP11B2CYP11B1RPS6KA5AGTR1AGTR2
SCHEMBL3065922 0.83 RPS6KA5 (0.42) CYP11B2CYP11B1RPS6KA5AGTR1AGTR2
SCHEMBL3049258 0.82 CYP11B1 (0.40) CYP11B2CYP11B1RPS6KA5NLRP3ALDH1A1
SCHEMBL3065402 0.82 TDP1 (0.42) CYP11B2CYP11B1NLRP3GAAPKM
SCHEMBL3064812 0.81 CYP11B1 (0.39) CYP11B2CYP11B1RPS6KA5AGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7300945-B2 Benzimidazole and pyridylimidazole derivatives NEUROGEN CORPORATION (US) 2007-11-27 US disclosed
US-20060025425-A1 Benzimidazole and pyridylimidazole derivatives NEUROGEN CORPORATION 2006-02-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060025425-A1 Benzimidazole and pyridylimidazole derivatives GABBR1, GABBR2, GABRA2 CYP11B2 47/4885CYP11B1 77/4885RPS6KA5 2860/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.