SCHEMBL5633461

SCHEMBL5633461

O=C(O)N1CCC(c2nnc(-c3ccccc3)o2)CC1

nearest known ligand 0.62

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.62
CYP2C9 P11712 1/20 0.62
HDAC1 Q13547 1/20 0.62
HDAC6 Q9UBN7 1/20 0.62
TNKS O95271 9/20 0.56
PARP1 P09874 9/20 0.56
PARP2 Q9UGN5 9/20 0.56
MAPT P10636 1/20 0.55
HSD11B1 P28845 1/20 0.53
POLB P06746 1/20 0.51
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
TP53 P04637 2/20 0.48
RXFP1 Q9HBX9 1/20 0.48
TSHR P16473 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14637530 0.88 MAPT (0.55) HDAC3CYP2C9HDAC1HDAC6TNKS
SCHEMBL22227916 0.83 MAPT (0.53) HDAC3CYP2C9HDAC1HDAC6TNKS
SCHEMBL22228020 0.83 MAPT (0.48) HDAC3CYP2C9HDAC1HDAC6TNKS
SCHEMBL440844 0.83 SMN1; SMN2 (0.65) HDAC3CYP2C9HDAC1HDAC6TNKS
SCHEMBL14638193 0.83 TNKS (0.54) HDAC3CYP2C9HDAC1HDAC6TNKS
SCHEMBL17339930 0.82 POLB (0.55) HDAC3CYP2C9HDAC1HDAC6TNKS
SCHEMBL462934 0.81 ALDH1A1 (0.52) HDAC3CYP2C9HDAC1HDAC6TNKS
SCHEMBL22227907 0.81 MAPT (0.47) HDAC3CYP2C9HDAC1HDAC6TNKS
SCHEMBL13666086 0.81 RBP4 (0.55) HDAC3CYP2C9HDAC1HDAC6TNKS
SCHEMBL16400168 0.80 LMNA (0.40) HDAC3CYP2C9HDAC1HDAC6TNKS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2731942-A1 NOVEL 2-PIPERIDIN-1-YL-ACETAMIDE COMPOUNDS FOR USE AS TANKYRASE INHIBITORS Novartis AG (CH) 2014-05-21 EP disclosed
US-7217714-B1 CCR5 modulators AGOURON PHARMACEUTICALS, INC. (US) 2007-05-15 US disclosed