SCHEMBL5636610

SCHEMBL5636610

C[Sn](C)(C)c1c(F)cccc1F

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.39
CES2 O00748 2/20 0.36
CES1 P23141 2/20 0.36
BCHE P06276 1/20 0.32
NFE2L2 Q16236 3/20 0.32
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
ALB P02768 1/20 0.30
ERN1 O75460 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5636759 0.83 TAAR1 (0.41) ALDH1A1SMN1; SMN2
SCHEMBL5702104 0.82 ACHE (0.39) ACHECES2CES1BCHENFE2L2
SCHEMBL5701891 0.71 RAPGEF4 (0.33) CES2CES1ALDH1A1ERN1
SCHEMBL5951408 0.70 CES2 (0.38) ACHECES2CES1BCHEKDM4E
SCHEMBL5702143 0.69 SMN1; SMN2 (0.36) ACHEKDM4ESMN1; SMN2
SCHEMBL5951303 0.69 ACHE (0.43) ACHECES2CES1NFE2L2ALDH1A1
SCHEMBL5637066 0.67 TSHR (0.35)
SCHEMBL2653065 0.65
SCHEMBL5638102 0.65 KIF11 (0.39) CES1KDM4EALDH1A1SMN1; SMN2
SCHEMBL254224 0.65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39679-E1 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2007-06-05 US disclosed
EP-1211256-B1 Method for purifying fluoroaryl metal compound NIPPON CATALYTIC CHEM IND (JP) 2006-08-02 EP disclosed
US-6713471-B1 SUCH AS TERT-BUTYL-1-METHYL-6,7,9,12-TETRAHYDRO-5H-PYRIDO-(4,3-B)(1,4) THIAZEPINO(2,3,4-HI)INDOLE-11(10H)-CARBOXYLATE; SEROTONIN AGONISTS AND ANTAGONISTS; CENTRAL NERVOUS SYSTEM DISORDERS BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-03-30 US disclosed
US-6509488-B2 Magnesium halide is precipitated and removed from solution containing fluoroaryl metal compound, magnesium halide, and ether solvent, or magnesium halide is removed by treating solution with acid NIPPON SHOKUBAI CO., LTD. (JP) 2003-01-21 US disclosed
EP-1211256-A2 Method for purifying fluoroaryl metal compound Nippon Shokubai Co., Ltd. (JP) 2002-06-05 EP disclosed
US-20020065425-A1 Method for purifying fluoroaryl metal compound NIPPON SHOKUBAI CO., LTD. (JP) 2002-05-30 US disclosed
EP-1192165-A2 SUBSTITUTED HETEROCYCLE FUSED GAMMA-CARBOLINES Bristol-Myers Squibb Pharma Company (US) 2002-04-03 EP disclosed
WO-2000077010-A2 SUBSTITUTED HETEROCYCLE FUSED GAMMA-CARBOLINES DU PONT PHARMACEUTICALS COMPANY (US) 2000-12-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020065425-A1 Method for purifying fluoroaryl metal compound MLLT3, AFF2, AFF4 ACHE 42/4885CES2 2108/4885CES1 2877/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.