SCHEMBL5648264

SCHEMBL5648264

CCN(CC)Cc1cnc2cc(N)c(OC)cc2c1

nearest known ligand 0.48

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PDGFRB P09619 13/20 0.48
PDGFRA P16234 13/20 0.48
EGFR P00533 1/20 0.39
PDE10A Q9Y233 3/20 0.39
ACHE P22303 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5644738 0.77 PDGFRB (0.42) PDGFRBPDGFRAACHE
SCHEMBL5645610 0.74 MCHR1 (0.45) PDGFRBPDGFRA
SCHEMBL5646416 0.73 PDGFRB (0.47) PDGFRBPDGFRA
SCHEMBL17450407 0.70 ALDH1A1 (0.62) ACHE
SCHEMBL12471340 0.69 PDE10A (0.47) PDE10A
Hydrochloric Acid SCHEMBL11277758 0.66 ACHE (0.51) ACHE
SCHEMBL29922921 0.65 NQO2 (0.56)
SCHEMBL5696548 0.65 NQO2 (0.56)
SCHEMBL3391498 0.65 PDGFRB (0.57) PDGFRBPDGFRA
SCHEMBL22185958 0.64 PDGFRB (0.50) PDGFRBPDGFRAEGFRPDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7183415-B2 Quinoline compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-02-27 US disclosed
US-7183415-B2 Quinoline compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-02-27 US disclosed
US-7183415-B2 Quinoline compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-02-27 US disclosed
US-20050209213-A1 Quinoline compound TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2005-09-22 US disclosed
EP-1447402-A1 QUINOLINE COMPOUND Takeda Chemical Industries, Ltd. (JP) 2004-08-18 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050209213-A1 Quinoline compound MC1R, MC2R, TYR PDGFRB 2194/4885PDGFRA 2217/4885EGFR 3760/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.