SCHEMBL5651048

SCHEMBL5651048

O=C(OC(=O)c1ccc(F)cc1F)c1ccc(F)cc1F

nearest known ligand 0.65

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CES2 O00748 3/20 0.65
CES1 P23141 3/20 0.65
RAB9A P51151 1/20 0.50
L3MBTL1 Q9Y468 2/20 0.49
MAPT P10636 3/20 0.48
POLB P06746 2/20 0.48
TDP1 Q9NUW8 1/20 0.48
ALDH1A1 P00352 2/20 0.47
GAA P10253 1/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
KLK7 P49862 1/20 0.43
SNCA P37840 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30954392 0.89 CES2 (0.68) CES2CES1RAB9AL3MBTL1MAPT
SCHEMBL23421455 0.88 CES2 (0.57) CES2CES1RAB9AL3MBTL1MAPT
SCHEMBL5651058 0.88 CES2 (0.52) CES2CES1RAB9AL3MBTL1MAPT
SCHEMBL8359445 0.87 CES2 (0.65) CES2CES1RAB9AL3MBTL1MAPT
SCHEMBL28305665 0.85 ALDH1A1 (0.49) CES2CES1RAB9AL3MBTL1MAPT
SCHEMBL523258 0.83 CES2 (0.61) CES2CES1RAB9AL3MBTL1MAPT
SCHEMBL14012584 0.83 CES2 (0.61) CES2CES1RAB9AL3MBTL1MAPT
SCHEMBL20551726 0.83 CES2 (0.61) CES2CES1RAB9AL3MBTL1MAPT
SCHEMBL6968044 0.83 CES2 (0.61) CES2CES1RAB9AL3MBTL1MAPT
SCHEMBL24779498 0.83 CES2 (0.61) CES2CES1RAB9AL3MBTL1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7235559-B1 Therapeutic quinazoline derivatives ASTRAZENECA AB (SE) 2007-06-26 US disclosed
EP-1218355-A1 THERAPEUTIC QUINAZOLINE DERIVATIVES AstraZeneca AB (SE) 2002-07-03 EP disclosed
WO-2001021597-A1 THERAPEUTIC QUINAZOLINE DERIVATIVES ASTRAZENECA AB (SE) 2001-03-29 WO disclosed
US-4255594-A Hydrogenation of halogen-containing carboxylic anhydrides ALLIED CHEMICAL CORPORATION (US) 1981-03-10 US disclosed