SCHEMBL5657660

SCHEMBL5657660

O=C(Cl)c1coc(Oc2cc(Cl)cc(Cl)c2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.42
MAPT P10636 4/20 0.42
NPSR1 Q6W5P4 4/20 0.41
KDM4E B2RXH2 2/20 0.34
GAA P10253 2/20 0.34
TPMT P51580 1/20 0.34
MEN1 O00255 1/20 0.33
GLA P06280 1/20 0.33
POLB P06746 1/20 0.33
CRHBP P24387 1/20 0.33
RECQL P46063 1/20 0.33
KMT2A Q03164 1/20 0.33
CRHR2 Q13324 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
MAPK1 P28482 1/20 0.32
MRGPRX4 Q96LA9 1/20 0.31
CARM1 Q86X55 1/20 0.30
PRMT6 Q96LA8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7074073 0.73 NR4A2 (0.38) ALDH1A1KDM4EGAATPMTMEN1
SCHEMBL7073706 0.70 GLRA1 (0.38) KDM4EPOLBMAPK1MRGPRX4
SCHEMBL93282 0.66 TPMT (0.62) TPMT
SCHEMBL6581228 0.66 MAPT (0.38) ALDH1A1MAPTNPSR1KMT2ACARM1
SCHEMBL11404150 0.66 AKR1C3 (0.53) KMT2A
SCHEMBL6633087 0.65 PARP10 (0.55) ALDH1A1MEN1KMT2A
Hydrochloric Acid SCHEMBL28632192 0.65 TPMT (0.59) GAATPMT
SCHEMBL6808605 0.64 ALDH1A1 (0.40) ALDH1A1MAPTNPSR1KDM4EGAA
SCHEMBL9357016 0.64 DAO (0.31) ALDH1A1MEN1POLBRECQLKMT2A
SCHEMBL10706723 0.63 TSHR (0.57) ALDH1A1MAPTTPMTKMT2ACARM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070043080-A1 Substituted anilinic piperidines as MCH selective antagonists MARZABADI MOHAMMAD R 2007-02-22 US disclosed
US-7067534-B1 Substituted anilinic piperidines as MCH selective antagonists H. LUNDBECK A/S (DK) 2006-06-27 US disclosed
US-6727264-B1 MELANIN CONCENTRATING HORMONE-1 RECEPTOR ANTAGONISTS; SLEEP, EATING, SEXUAL DISORDERS SYNAPTIC PHARMACEUTICAL CORPORATION 2004-04-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070043080-A1 Substituted anilinic piperidines as MCH selective antagonists MCHR1, MCHR2, MC1R ALDH1A1 620/4885MAPT 2336/4885NPSR1 19/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.