SCHEMBL5657750

SCHEMBL5657750

[CH2]C(CN)Cc1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 2/20 0.52
TAAR1 Q96RJ0 4/20 0.48
SLC6A2 P23975 2/20 0.48
CYP2A6 P11509 2/20 0.48
MAOA P21397 1/20 0.48
SLC6A4 P31645 1/20 0.48
SLC6A3 Q01959 1/20 0.48
SIGMAR1 Q99720 1/20 0.48
ADORA2A P29274 1/20 0.48
ADORA1 P30542 1/20 0.48
LOXL2 Q9Y4K0 2/20 0.46
ANPEP P15144 1/20 0.45
CYP2D6 P10635 1/20 0.45
ALPI P09923 1/20 0.43
PKM P14618 1/20 0.43
PTGS1 P23219 1/20 0.43
XIAP P98170 1/20 0.43
SLC7A5 Q01650 1/20 0.43
HTR2A P28223 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1287678 0.85 EPHX1 (0.55) EPHX1TAAR1SLC6A2CYP2A6MAOA
SCHEMBL523308 0.78 EPHX1 (0.48) EPHX1TAAR1SLC6A2CYP2A6MAOA
SCHEMBL8780026 0.76 TRPA1 (0.54) EPHX1TAAR1SLC6A2CYP2A6MAOA
SCHEMBL8660787 0.76 EPHX1 (0.46) EPHX1TAAR1SLC6A2CYP2A6MAOA
SCHEMBL1376582 0.76 TRPA1 (0.50) EPHX1TAAR1SLC6A2CYP2A6MAOA
SCHEMBL516032 0.75 EPHX1 (0.56) EPHX1TAAR1SLC6A2CYP2A6MAOA
SCHEMBL6563096 0.75 EPHX1 (0.56) EPHX1TAAR1SLC6A2CYP2A6MAOA
SCHEMBL351709 0.75 EPHX1 (0.64) EPHX1TAAR1SLC6A2CYP2A6MAOA
SCHEMBL1007428 0.75 EPHX1 (0.50) EPHX1TAAR1SLC6A2CYP2A6MAOA
SCHEMBL6931237 0.75 EPHX1 (0.64) EPHX1TAAR1SLC6A2CYP2A6MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1863530-A (3,4-phenyl)piperidin-3-yl- phenylcarboxylate derivatives and related compounds as beta-secretase inhibitors for the treatment of alzheimer's disease ELAN PHARM INC (US) 2006-11-15 CN claimed
CN-104145212-A Composition for forming liquid crystal alighment film and liquid crystal display element SOKI CORP 2014-11-12 CN disclosed
CN-101914040-A Acyloxyalkyl carbamate prodrugs, synthetic method and purposes XENOPORT INC 2010-12-15 CN disclosed
CN-1860101-B Acyloxyalkyl carbamate prodrugs, synthesis methods and uses XENOPORT INC 2010-10-27 CN disclosed
CN-101001612-A Controlled release dosage forms for gamma aminobutyric acid receptor agonists IMPAX LABORATORIES INC (US) 2007-07-18 CN disclosed
CN-1863530-A (3,4-phenyl)piperidin-3-yl- phenylcarboxylate derivatives and related compounds as beta-secretase inhibitors for the treatment of alzheimer's disease ELAN PHARM INC (US) 2006-11-15 CN disclosed
CN-1860101-A Acyloxyalkyl carbamate prodrugs, synthesis methods and uses XENOPORT INC (US) 2006-11-08 CN disclosed
EP-1401423-A4 METHOD OF TREATING GASTROESOPHAGEAL REFLUX DISEASE AND NOCTURNAL ACID BREAKTHROUGH DEPOMED DEV LTD (BM) 2006-08-16 EP disclosed
EP-1401423-A1 METHOD OF TREATING GASTROESOPHAGEAL REFLUX DISEASE AND NOCTURNAL ACID BREAKTHROUGH Depomed Development, Ltd (GB) 2004-03-31 EP disclosed
CN-1117560-C Reflux inhibitors ASTRA AB (SE) 2003-08-13 CN disclosed
US-20030031711-A1 Method of treating gastroesophageal reflux disease and nocturnal acid breakthrough ASSERTIO THERAPEUTICS, INC. 2003-02-13 US disclosed
WO-2002096404-A1 METHOD OF TREATING GASTROESOPHAGEAL REFLUX DISEASE AND NOCTURNAL ACID BREAKTHROUGH DEPOMED DEVELOPMENT LTD (GB) 2002-12-05 WO disclosed
CN-1237105-A Reflux inhibitors ASTRA AB (SE) 1999-12-01 CN disclosed