SCHEMBL5658074

SCHEMBL5658074

Nc1nc(SCC(=O)NCc2ccccc2)ncc1C(=O)O

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.61
GLA P06280 2/20 0.59
LMNA P02545 2/20 0.59
GAA P10253 1/20 0.56
MAPK1 P28482 2/20 0.53
NPSR1 Q6W5P4 1/20 0.51
SMN1; SMN2 Q16637 4/20 0.50
NPC1 O15118 3/20 0.50
RAB9A P51151 3/20 0.50
TSHR P16473 2/20 0.50
KDM4E B2RXH2 2/20 0.50
NFKB1 P19838 1/20 0.50
NFKB2 Q00653 1/20 0.50
RELA Q04206 1/20 0.50
MAPK10 P53779 1/20 0.50
POLB P06746 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2D6 P10635 1/20 0.49
MAPT P10636 1/20 0.49
CYP2C9 P11712 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5120763 0.81 SMN1; SMN2 (0.71) ALDH1A1LMNAGAASMN1; SMN2NPC1
SCHEMBL5660091 0.80 RAB9A (0.47) ALDH1A1GLALMNAGAAMAPK1
SCHEMBL5659327 0.73 ALDH1A1 (0.52) ALDH1A1LMNAGAAMAPK1SMN1; SMN2
SCHEMBL5658477 0.73 ALDH1A1 (0.57) ALDH1A1LMNAMAPK1SMN1; SMN2NPC1
SCHEMBL5659351 0.73 ALDH1A1 (0.49) ALDH1A1LMNAMAPK1SMN1; SMN2NPC1
SCHEMBL1158167 0.72 SMN1; SMN2 (0.52) ALDH1A1LMNAMAPK1SMN1; SMN2NPC1
SCHEMBL12961782 0.70 ALDH1A1 (0.79) ALDH1A1LMNAGAASMN1; SMN2NPC1
SCHEMBL5658070 0.70 SMN1; SMN2 (0.46) ALDH1A1LMNAGAASMN1; SMN2NPC1
SCHEMBL5726116 0.69 ALDH1A1 (0.48) ALDH1A1GAAMAPK1SMN1; SMN2NPC1
SCHEMBL24846493 0.68 ENPP1 (0.73) ALDH1A1GLALMNAGAASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7176310-B1 Pyrimidinecarboxamide derivatives and their use as anti-inflammatory agents UCB SA (GB) 2007-02-13 US disclosed