SCHEMBL56582

SCHEMBL56582

Cc1c(OP(=O)(O)CCC(NC(=O)OCc2ccccc2)C(=O)OCc2ccccc2)cccc1[N+](=O)[O-]

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
CYP1A2 P05177 1/20 0.43
POLB P06746 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C19 P33261 1/20 0.43
GSTP1 P09211 1/20 0.42
GSTM2 P28161 1/20 0.42
CTSL P07711 8/20 0.42
CTSB P07858 8/20 0.42
HDAC1 Q13547 2/20 0.42
HDAC2 Q92769 2/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
KYNU Q16719 1/20 0.41
ELANE P08246 1/20 0.40
ALOX15 P16050 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL56757 0.86 HDAC1 (0.51) CTSLCTSBHDAC1HDAC2
SCHEMBL56738 0.83 HDAC1 (0.46) CTSLCTSBHDAC1HDAC2MEN1
SCHEMBL56407 0.79 OPRK1 (0.44) POLBCTSLKYNUELANE
SCHEMBL21174053 0.77 KYNU (0.58) ALDH1A1CTSLCTSBKYNUELANE
SCHEMBL21189192 0.77 KYNU (0.58) ALDH1A1CTSLCTSBKYNUELANE
SCHEMBL13774904 0.77 GRM8 (0.55) ALDH1A1CYP1A2POLBCYP3A4CYP2C19
SCHEMBL57018 0.77 CTSL (0.48) CTSLKYNUELANE
SCHEMBL56832 0.76 HDAC1 (0.53) CTSLHDAC1HDAC2
SCHEMBL56509 0.76 GRM8 (0.57)
SCHEMBL56919 0.76 CTSL (0.43) CTSLKYNUELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129557-B2 Phosphonic acid diester derivative and method for producing thereof Nagai, Kazuhiro (JP) 2012-03-06 US disclosed
US-20090163725-A1 PHOSPHONIC ACID DIESTER DERIVATIVE AND METHOD FOR PRODUCING THEREOF HIRATAKE, GOU (JP) 2009-06-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090163725-A1 PHOSPHONIC ACID DIESTER DERIVATIVE AND METHOD FOR PRODUCING THEREOF PPA1, G6PD, PHOSPHO1 ALDH1A1 1716/4885CYP1A2 1147/4885POLB 841/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.