SCHEMBL5658453

SCHEMBL5658453

NC(=O)N1CCC(C2CCN(C(=O)[CH]Cc3cc(Br)c4[nH]ncc4c3)CC2)CC1

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CALCA P06881 7/20 0.33
ROCK2 O75116 4/20 0.32
CYP3A4 P08684 3/20 0.32
CALCRL Q16602 2/20 0.32
BTK Q06187 1/20 0.31
FNTA P49354 4/20 0.31
FNTB P49356 4/20 0.31
HRAS P01112 1/20 0.31
KRAS P01116 1/20 0.31
ABCB1 P08183 1/20 0.31
PAK1 Q13153 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5657191 0.91 CALCA (0.40) CALCA
SCHEMBL5661443 0.91 CALCA (0.40) CALCA
SCHEMBL5660254 0.88 CYP3A4 (0.36) CALCAROCK2CYP3A4CALCRLBTK
SCHEMBL5659680 0.87 CYP3A4 (0.37) CALCAROCK2CYP3A4CALCRLBTK
SCHEMBL5657726 0.85 RXRA (0.40) CALCAROCK2CYP3A4BTKPAK1
SCHEMBL5660671 0.82 ROCK2 (0.44) ROCK2CYP3A4
SCHEMBL5658727 0.80 BTK (0.36) ROCK2CYP3A4BTK
SCHEMBL5659437 0.80 BTK (0.36) ROCK2CYP3A4CALCRLBTK
SCHEMBL4862072 0.80 ACACB (0.38) CALCA
SCHEMBL5661661 0.79 CALCA (0.47) CALCACALCRL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050227968-A1 Selected CGRP-antagonists process for preparing them and their use as pharmaceutical compositions BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2005-10-13 US claimed
US-7205294-B2 Selected CGRP-antagonists process for preparing them and their use as pharmaceutical compositions BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-04-17 US disclosed
US-20050227968-A1 Selected CGRP-antagonists process for preparing them and their use as pharmaceutical compositions BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2005-10-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050227968-A1 Selected CGRP-antagonists process for preparing them and their use as pharmaceutical compositions BDKRB1, BDKRB2, CALCRL CALCA 7/4885ROCK2 4518/4885CYP3A4 1053/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.