SCHEMBL5660734

SCHEMBL5660734

CC1(C)OC(=O)N(C(=O)O)C1c1ccc(F)c(F)c1

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 1/20 0.39
HCAR2 Q8TDS4 1/20 0.39
HTR7 P34969 1/20 0.36
TNKS O95271 10/20 0.35
TSHR P16473 1/20 0.34
HSD11B1 P28845 1/20 0.32
CCR2 P41597 1/20 0.32
ADRA1A P35348 4/20 0.32
ADRA1B P35368 4/20 0.32
ADRA1D P25100 3/20 0.32
HRH1 P35367 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14587408 0.89 HCAR3 (0.36) HCAR3HCAR2HTR7TNKSTSHR
SCHEMBL14619731 0.84 TNKS (0.37) HCAR3HCAR2TNKS
SCHEMBL7840377 0.81 HTR7 (0.36) HCAR3HCAR2HTR7TSHRCCR2
SCHEMBL7095750 0.71 ADRA1A (0.52) HCAR3HCAR2HTR7TSHRADRA1A
SCHEMBL6082094 0.71 ADRA1A (0.52) HCAR3HCAR2HTR7TSHRADRA1A
SCHEMBL6959819 0.71 ADRA1A (0.52) HCAR3HCAR2HTR7TSHRADRA1A
SCHEMBL6964542 0.70 TNKS (0.32) HCAR3HCAR2TNKSADRA1AADRA1B
SCHEMBL6227914 0.69 MTOR (0.37) HTR7TSHRADRA1AADRA1BADRA1D
SCHEMBL6082708 0.69 MTOR (0.37) HTR7TSHRADRA1AADRA1BADRA1D
SCHEMBL5660885 0.69 MTOR (0.37) HTR7TSHRADRA1AADRA1BADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070043080-A1 Substituted anilinic piperidines as MCH selective antagonists MARZABADI MOHAMMAD R 2007-02-22 US disclosed
US-7067534-B1 Substituted anilinic piperidines as MCH selective antagonists H. LUNDBECK A/S (DK) 2006-06-27 US disclosed
US-6727264-B1 MELANIN CONCENTRATING HORMONE-1 RECEPTOR ANTAGONISTS; SLEEP, EATING, SEXUAL DISORDERS SYNAPTIC PHARMACEUTICAL CORPORATION 2004-04-27 US disclosed
US-20040038855-A1 DNA encoding a human melanin concentrating hormone receptor (MCH1) and uses thereof H. LUNDBECK A/S (DK) 2004-02-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070043080-A1 Substituted anilinic piperidines as MCH selective antagonists MCHR1, MCHR2, MC1R HCAR3 83/4885HCAR2 73/4885HTR7 128/4885
US-20040038855-A1 DNA encoding a human melanin concentrating hormone receptor (MCH1) and uses thereof MCHR1, MCHR2, MC1R HCAR3 69/4885HCAR2 191/4885HTR7 217/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.