SCHEMBL5665659

SCHEMBL5665659

COc1cccc(B(O)ON)c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 2/20 0.67
PRSS1 P07477 1/20 0.49
PRSS2 P07478 1/20 0.49
PRSS3 P35030 1/20 0.49
ALDH1A1 P00352 1/20 0.47
CYP3A4 P08684 1/20 0.47
IDO1 P14902 2/20 0.44
AGXT P21549 2/20 0.44
PARP1 P09874 1/20 0.44
CA1 P00915 2/20 0.44
CA2 P00918 2/20 0.44
ACHE P22303 1/20 0.44
HTR3E A5X5Y0 1/20 0.43
HTR3B O95264 1/20 0.43
HTR3A P46098 1/20 0.43
HTR3D Q70Z44 1/20 0.43
HTR3C Q8WXA8 1/20 0.43
CES2 O00748 1/20 0.43
CES1 P23141 1/20 0.43
CA7 P43166 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28329900 0.81 ENPP2 (0.67) ENPP2PRSS1PRSS2PRSS3ALDH1A1
SCHEMBL28041771 0.81 ENPP2 (0.67) ENPP2PRSS1PRSS2PRSS3ALDH1A1
SCHEMBL480132 0.81 ENPP2 (0.67) ENPP2PRSS1PRSS2PRSS3ALDH1A1
SCHEMBL27951222 0.81 ENPP2 (0.67) ENPP2PRSS1PRSS2PRSS3ALDH1A1
SCHEMBL7344145 0.80 ENPP2 (1.00) ENPP2PRSS1PRSS2PRSS3ALDH1A1
SCHEMBL5140 0.80 ENPP2 (1.00) ENPP2PRSS1PRSS2PRSS3ALDH1A1
SCHEMBL5665675 0.80 CA1 (0.61) ENPP2PRSS1PRSS2PRSS3ALDH1A1
SCHEMBL7344156 0.80 ENPP2 (0.65) ENPP2PRSS1PRSS2PRSS3ALDH1A1
Methyl Alcohol SCHEMBL28712606 0.79 ENPP2 (0.96) ENPP2PRSS1PRSS2PRSS3ALDH1A1
SCHEMBL12524808 0.79 ENPP2 (0.74) ENPP2PRSS1PRSS2PRSS3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730118-A1 SUBSTITUTED AZOLE DERIVATIVES, COMPOSITIONS, AND METHODS OF USE Transtech Pharma, Inc. (US) 2006-12-13 EP disclosed
WO-2005080346-A1 SUBSTITUTED AZOLE DERIVATIVES, COMPOSITIONS, AND METHODS OF USE TRANSTECH PHARMA, INC. (US) 2005-09-01 WO disclosed