SCHEMBL7344156

SCHEMBL7344156

COc1cccc(B(O)OB(OB(O)c2cccc(OC)c2)c2cccc(OC)c2)c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 2/20 0.65
CA1 P00915 2/20 0.46
CA2 P00918 2/20 0.46
CA7 P43166 1/20 0.46
CA9 Q16790 1/20 0.46
PRSS1 P07477 1/20 0.43
PRSS2 P07478 1/20 0.43
PRSS3 P35030 1/20 0.43
ACHE P22303 1/20 0.42
CES2 O00748 1/20 0.42
CES1 P23141 1/20 0.42
ALDH1A1 P00352 2/20 0.41
CYP3A4 P08684 1/20 0.41
CA4 P22748 1/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
PARP1 P09874 1/20 0.40
RELA Q04206 1/20 0.40
HTR3E A5X5Y0 1/20 0.39
HTR3B O95264 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4974695 0.91 ENPP2 (0.54) ENPP2CA1CA2CA7CA9
SCHEMBL27951222 0.80 ENPP2 (0.67) ENPP2CA1CA2CA7CA9
SCHEMBL28329900 0.80 ENPP2 (0.67) ENPP2CA1CA2CA7CA9
SCHEMBL28041771 0.80 ENPP2 (0.67) ENPP2CA1CA2CA7CA9
SCHEMBL480132 0.80 ENPP2 (0.67) ENPP2CA1CA2CA7CA9
SCHEMBL5665659 0.80 ENPP2 (0.67) ENPP2CA1CA2CA7CA9
SCHEMBL14986000 0.79 ENPP2 (0.64) ENPP2CA1CA2CA7CA9
SCHEMBL5140 0.79 ENPP2 (1.00) ENPP2CA1CA2CA7CA9
SCHEMBL7344145 0.79 ENPP2 (1.00) ENPP2CA1CA2CA7CA9
SCHEMBL26693034 0.78 ENPP2 (0.54) ENPP2CA1CA2PRSS1PRSS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0819125-A1 THIENYL-, FURYL-, PYRROLYL- AND BIPHENYLSULFONAMIDES AND DERIVATIVES THEREOF THAT MODULATE THE ACTIVITY OF ENDOTHELIN TEXAS BIOTECHNOLOGY CORPORATION (US) 1998-01-21 EP disclosed
WO-1996031492-A1 THIENYL-, FURYL-, PYRROLYL- AND BIPHENYLSULFONAMIDES AND DERIVATIVES THEREOF THAT MODULATE THE ACTIVITY OF ENDOTHELIN TEXAS BIOTECHNOLOGY CORPORATION (US) 1996-10-10 WO disclosed