SCHEMBL5671522

SCHEMBL5671522

NC(=O)c1ccc(F)c(F)c1CC1CCC(N)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 2/20 0.42
PARP10 Q53GL7 2/20 0.39
PARP15 Q460N3 1/20 0.39
BTK Q06187 5/20 0.36
ROCK1 Q13464 1/20 0.35
CES2 O00748 2/20 0.35
CES1 P23141 2/20 0.35
MAP2K2 P36507 2/20 0.34
MAP2K1 Q02750 2/20 0.34
RAF1 P04049 1/20 0.34
PDGFRB P09619 1/20 0.34
CSNK2A2 P19784 1/20 0.34
CSNK2B P67870 1/20 0.34
CSNK2A1 P68400 1/20 0.34
CSNK2A3 Q8NEV1 1/20 0.34
AURKC Q9UQB9 1/20 0.34
CAMK2A Q9UQM7 1/20 0.34
DGAT1 O75907 1/20 0.34
HTR1A P08908 1/20 0.34
JAK2 O60674 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6466321 0.75 ROCK2 (0.44) ROCK2PARP10PARP15ROCK1CES2
SCHEMBL6466316 0.75 ROCK2 (0.44) ROCK2PARP10PARP15ROCK1CES2
SCHEMBL28871862 0.73 KDM4E (0.41) PARP10PARP15
SCHEMBL2721695 0.70 PARP10 (0.56) PARP10PARP15CES2CES1MAP2K2
SCHEMBL5670138 0.69 PARP10 (0.39) PARP10PARP15CES2CES1MAP2K2
SCHEMBL8957045 0.68 ALDH1A1 (0.40) PARP10PARP15CYP2C9CYP2C19
SCHEMBL4552089 0.68 ROCK2 (0.39) ROCK2BTKCES2
SCHEMBL4552088 0.68 ROCK2 (0.39) ROCK2BTKCES2
SCHEMBL2770591 0.67 CES2 (0.42) ROCK2PARP10PARP15CES2CES1
SCHEMBL11162291 0.67 KDM4E (0.42) ROCK2PARP10PARP15BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730122-A2 PYRIMIDINE DERIVATIVES AND METHODS OF TREATMENT RELATED TO THE USE THEREOF TAISHO PHARMACEUTICAL CO., LTD (JP) 2006-12-13 EP disclosed
WO-2005095357-A2 PYRIMIDINE DERIVATIVES AND METHODS OF TREATMENT RELATED TO THE USE THEREOF TAISHO PHARMACEUTICAL CO., LTD. (JP) 2005-10-13 WO disclosed