SCHEMBL5673146

SCHEMBL5673146

CCc1cccc2cc(C)[nH]c12

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DAO P14920 4/20 0.60
FLT3 P36888 1/20 0.48
KDM4E B2RXH2 7/20 0.43
GAA P10253 2/20 0.43
ALDH1A1 P00352 6/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
HPGD P15428 2/20 0.41
HTT P42858 1/20 0.41
MAPT P10636 4/20 0.40
LMNA P02545 3/20 0.40
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
ALOX12 P18054 1/20 0.40
GABRA1 P14867 2/20 0.39
GABRB2 P47870 2/20 0.39
DDO Q99489 2/20 0.39
HSD17B10 Q99714 2/20 0.38
NPSR1 Q6W5P4 1/20 0.38
POLB P06746 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30548030 0.79 DAO (0.58) DAOFLT3KDM4EALDH1A1HPGD
SCHEMBL11386139 0.79 DAO (0.68) DAOFLT3KDM4EALDH1A1HPGD
SCHEMBL19708446 0.77 DAO (0.55) DAOFLT3KDM4EALDH1A1HPGD
SCHEMBL30712834 0.75 DAO (0.56) DAOKDM4EGAAALDH1A1SMN1; SMN2
SCHEMBL1093711 0.75 DAO (0.56) DAOKDM4EGAAALDH1A1SMN1; SMN2
SCHEMBL11658287 0.75 DHODH (0.55) DAOFLT3KDM4EALDH1A1SMN1; SMN2
SCHEMBL16767845 0.75 DAO (1.00) DAOFLT3KDM4EALDH1A1HPGD
SCHEMBL4048274 0.75 FLT3 (0.60) DAOFLT3KDM4EALDH1A1HPGD
SCHEMBL6135945 0.75 DAO (0.37) DAOFLT3KDM4EGAAALDH1A1
SCHEMBL4045458 0.74 RAB9A (0.59) DAOFLT3KDM4EGAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023078398-A1 COMPOUNDS AS BCL-2 INHIBITORS FOCHON PHARMACEUTICALS, LTD. (CN) 2023-05-11 WO disclosed
EP-1718608-B1 VIRAL POLYMERASE INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2013-07-17 EP disclosed
US-6995184-B2 Such as (7-chloro-2-methyl-1-(3-(methylsulphanyl)propyl)-1H-indol-3-yl)(2,3-dichloro-phenyl)methanone; cannabinoid receptors (cb2); G proteins coupled receptors SANOFI-AVENTIS (FR) 2006-02-07 US disclosed
CN-1234688-C 3-aroyl indoles and their use as CB2Use of receptor agonists SANOFI ANVANT (FR) 2006-01-04 CN disclosed
EP-1339679-B1 3-ARYLINDOLE DERIVATIVES AND THEIR USE AS CB2 RECEPTOR AGONISTS SANOFI AVENTIS (FR) 2005-08-10 EP disclosed
CN-1483023-A 3-arylindole derivatives and their use as cb2 receptor agonists ʥŵ��-�ϳ�ʵ���ҹ�˾ 2004-03-17 CN disclosed
US-20040034090-A1 3-Arylindole derivatives and their use as cb2 receptor agonists SANOFI-AVENTIS (FR) 2004-02-19 US disclosed
EP-1339679-A1 3-ARYLINDOLE DERIVATIVES AND THEIR USE AS CB2 RECEPTOR AGONISTS Sanofi-Aventis (FR) 2003-09-03 EP disclosed
WO-2002042269-A1 3-ARYLINDOLE DERIVATIVES AND THEIR USE AS CB2 RECEPTOR AGONISTS SANOFI-SYNTHELABO (FR) 2002-05-30 WO disclosed
US-RE29834-E PREPARED FROM 4-SULFONYL-1,8-NAPHTHOLACTAMS BAYER AKTIENGESELLSCHAFT (DE) 1978-11-14 US disclosed
US-3959310-A BENZINDOLE BAYER AKTIENGESELLSCHAFT (DT) 1976-05-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040034090-A1 3-Arylindole derivatives and their use as cb2 receptor agonists CNR2, CNR1, GPR52 DAO 2722/4885FLT3 1282/4885KDM4E 2393/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.