SCHEMBL5684774

SCHEMBL5684774

CCO[Si](CCCNc1ccc(C)cc1)(OCC)OCC

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.52
HRH3 Q9Y5N1 1/20 0.39
PTPN1 P18031 1/20 0.39
GAA P10253 5/20 0.36
ALDH1A1 P00352 4/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
HTT P42858 1/20 0.36
KDM4E B2RXH2 2/20 0.34
LMNA P02545 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
ACKR3 P25106 1/20 0.34
POLB P06746 1/20 0.34
HSP90AA1 P07900 1/20 0.34
HSP90AB1 P08238 1/20 0.34
THRB P10828 1/20 0.34
HPGD P15428 1/20 0.34
ALOX15 P16050 1/20 0.34
MAPK1 P28482 1/20 0.34
CASP1 P29466 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2763548 0.90 MAPT (0.55) MAPTHRH3PTPN1GAAALDH1A1
SCHEMBL5685426 0.85 MAPT (0.42) MAPTGAAALDH1A1MEN1KMT2A
SCHEMBL134305 0.85 ALDH1A1 (0.53) MAPTHRH3ALDH1A1KMT2ASMN1; SMN2
SCHEMBL3198023 0.84 GAA (0.58) MAPTPTPN1GAAALDH1A1MEN1
Hydrochloric Acid SCHEMBL29522911 0.83 ALDH1A1 (0.52) MAPTHRH3ALDH1A1SMN1; SMN2L3MBTL1
SCHEMBL5685420 0.83 MAPT (0.55) MAPTHRH3PTPN1GAAALDH1A1
SCHEMBL2116813 0.80 ALDH1A1 (0.52) MAPTALDH1A1HTTL3MBTL1
SCHEMBL16147721 0.80 MAPT (0.47) MAPTGAAALDH1A1L3MBTL1
SCHEMBL6441905 0.80 ALDH1A1 (0.47) MAPTALDH1A1MEN1KMT2AL3MBTL1
SCHEMBL4738119 0.80 ALDH1A1 (0.52) MAPTALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1478651-B1 PREPARATION OF N-SUBSTITUTED AMINOORGANOSILANES GEN ELECTRIC (US) 2006-02-08 EP claimed
EP-1478651-A1 PREPARATION OF N-SUBSTITUTED AMINOORGANOSILANES GENERAL ELECTRIC COMPANY (US) 2004-11-24 EP claimed
WO-2003070734-A1 PREPARATION OF N-SUBSTITUTED AMINOORGANOSILANES GENERAL ELECTRIC COMPANY (US) 2003-08-28 WO claimed
US-6448425-B1 N-CYCLOALKYLAMINOALKYLSILANES BY HYDROGENATING N-ARYLAMINO-ALKYLSILANES; PALLADIUM, PLATINUM, NICKEL, RHENIUM, RHODIUM, RUTHENIUM, COPPER CHROMITE CATALYST; N-CYCLOHEXYL-3-AMINOPROPYLTRIMETHOXYSILANE FROM CROMPTON CORPORATION 2002-09-10 US claimed
US-5530082-A DRY STORAGE STABLE MIXTURE OF POLYSILOXANE WHICH CURES TO ELASTOMER WITH MOISTURE AT ROOM TEMPERATURE, SILANE CROSSLINKING AGENT, ORGANIC TITANIUM CATALYST AND ADHESION PROMOTER BAYER AKTIENGESELLSCHAFT (DE) 1996-06-25 US claimed
EP-1478651-B1 PREPARATION OF N-SUBSTITUTED AMINOORGANOSILANES GEN ELECTRIC (US) 2006-02-08 EP disclosed
EP-1478651-A1 PREPARATION OF N-SUBSTITUTED AMINOORGANOSILANES GENERAL ELECTRIC COMPANY (US) 2004-11-24 EP disclosed
WO-2003070734-A1 PREPARATION OF N-SUBSTITUTED AMINOORGANOSILANES GENERAL ELECTRIC COMPANY (US) 2003-08-28 WO disclosed
US-6448425-B1 N-CYCLOALKYLAMINOALKYLSILANES BY HYDROGENATING N-ARYLAMINO-ALKYLSILANES; PALLADIUM, PLATINUM, NICKEL, RHENIUM, RHODIUM, RUTHENIUM, COPPER CHROMITE CATALYST; N-CYCLOHEXYL-3-AMINOPROPYLTRIMETHOXYSILANE FROM CROMPTON CORPORATION 2002-09-10 US disclosed
US-5530082-A DRY STORAGE STABLE MIXTURE OF POLYSILOXANE WHICH CURES TO ELASTOMER WITH MOISTURE AT ROOM TEMPERATURE, SILANE CROSSLINKING AGENT, ORGANIC TITANIUM CATALYST AND ADHESION PROMOTER BAYER AKTIENGESELLSCHAFT (DE) 1996-06-25 US disclosed