SCHEMBL5685667

SCHEMBL5685667

CNS(=O)(=O)c1ccc(Cc2ccccc2C(N)=O)cc1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.52
CA2 P00918 2/20 0.52
CA9 Q16790 1/20 0.52
IKBKB O14920 1/20 0.49
CHUK O15111 1/20 0.49
TSHR P16473 1/20 0.44
L3MBTL1 Q9Y468 2/20 0.43
GAA P10253 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
NPC1 O15118 1/20 0.41
HPGD P15428 1/20 0.41
RAB9A P51151 1/20 0.41
NR3C2 P08235 1/20 0.41
KDM1A O60341 1/20 0.40
MAOA P21397 1/20 0.40
ANXA2 P07355 1/20 0.40
S100A10 P60903 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL933463 0.85 CA1 (0.55) CA1CA2CA9IKBKBCHUK
SCHEMBL5682926 0.85 L3MBTL1 (0.44) CA1CA2CA9IKBKBCHUK
SCHEMBL5677878 0.84 CA2 (0.72) CA1CA2CA9TSHRSMN1; SMN2
SCHEMBL30100451 0.79 TSHR (0.51) CA1CA2CA9TSHRGAA
SCHEMBL1004028 0.78 TSHR (0.58) CA1CA2CA9TSHRKDM4E
SCHEMBL19439093 0.77 TSHR (0.53) CA1CA2CA9TSHRKDM4E
SCHEMBL5723934 0.77 KEAP1 (0.56) CA1CA2CA9TSHRKDM4E
SCHEMBL9367212 0.77 TSHR (0.54) CA1CA2CA9TSHRNPC1
Hydrochloric Acid SCHEMBL15690391 0.76 TSHR (0.56) CA1CA2CA9TSHRKDM4E
SCHEMBL1500536 0.75 TSHR (0.51) CA1CA2CA9TSHRSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1633714-A1 2-AMINO-PYRIDINE DERIVATIVES AS BETA-2 ADRENORECEPTOR AGONISTS Pfizer Limited (GB) 2006-03-15 EP disclosed
WO-2004108675-A1 2-AMINO-PYRIDINE DERIVATIVES AS BETA-2 ADRENORECEPTOR AGONISTS PFIZER LIMITED (GB) 2004-12-16 WO disclosed