SCHEMBL5686103

SCHEMBL5686103

CCOC(=O)CC(C)(C)/C=C/C(Cl)(Br)C(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MGAM O43451 1/20 0.33
GAA P10253 1/20 0.33
SI P14410 1/20 0.33
MGAM2 Q2M2H8 1/20 0.33
HSD11B1 P28845 1/20 0.33
GSK3A P49840 1/20 0.32
GSK3B P49841 1/20 0.32
POLB P06746 2/20 0.31
NPSR1 Q6W5P4 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.30
PTP4A1 Q93096 1/20 0.30
PDK1 Q15118 1/20 0.30
PDK2 Q15119 1/20 0.30
PDK3 Q15120 1/20 0.30
PDK4 Q16654 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5686106 1.00 TRPA1 (0.35) TRPA1ALDH1A1MGAMGAASI
SCHEMBL11030953 0.84 ALDH1A1 (0.37) TRPA1ALDH1A1MGAMGAASI
SCHEMBL11027583 0.84 ALDH1A1 (0.37) TRPA1ALDH1A1MGAMGAASI
SCHEMBL5683340 0.84 GAA (0.35) TRPA1ALDH1A1MGAMGAASI
SCHEMBL5683344 0.84 GAA (0.35) TRPA1ALDH1A1MGAMGAASI
SCHEMBL5686096 0.84
SCHEMBL5686092 0.84
SCHEMBL9796681 0.80 GAA (0.40) TRPA1ALDH1A1MGAMGAASI
SCHEMBL9796686 0.80 GAA (0.40) TRPA1ALDH1A1MGAMGAASI
SCHEMBL8406765 0.79 HMGCR (0.34) CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832873-B1 Preparation of cyclopropane esters SYNGENTA LTD (GB) 2006-03-08 EP disclosed
EP-0793638-B1 PREPARATION OF CYCLOPROPANE ESTERS ZENECA LTD (GB) 1999-06-30 EP disclosed
EP-0700375-B1 PREPARATION OF CYCLOPROPANE ESTERS ZENECA LTD (GB) 1998-12-23 EP disclosed
EP-0700373-B1 PREPARATION OF HALOGENATED ALCOHOLS ZENECA LTD (GB) 1998-04-22 EP disclosed
EP-0832873-A1 Preparation of cyclopropane esters ZENECA LIMITED (GB) 1998-04-01 EP disclosed
US-5731475-A Preparation of cyclopropane esters ZENECA LIMITED (GB) 1998-03-24 US disclosed
US-5723649-A Preparation of cyclopropane esters ZENECA LIMITED (GB) 1998-03-03 US disclosed
US-5670697-A Preparation of cyclopropane esters ZENECA LIMITED (GB) 1997-09-23 US disclosed
EP-0793638-A1 PREPARATION OF CYCLOPROPANE ESTERS ZENECA LIMITED (GB) 1997-09-10 EP disclosed
US-5527972-A Preparation and use of halogenated alcohols ZENECA LIMITED (GB) 1996-06-18 US disclosed
WO-1996016018-A1 PREPARATION OF CYCLOPROPANE ESTERS ZENECA LIMITED (GB) 1996-05-30 WO disclosed
EP-0700375-A1 PREPARATION OF CYCLOPROPANE ESTERS ZENECA LIMITED (GB) 1996-03-13 EP disclosed
EP-0700373-A1 PREPARATION OF HALOGENATED ALCOHOLS ZENECA LIMITED (GB) 1996-03-13 EP disclosed
WO-1994027951-A1 PREPARATION OF CYCLOPROPANE ESTERS ZENECA LIMITED (GB) 1994-12-08 WO disclosed
WO-1994027942-A1 PREPARATION OF HALOGENATED ALCOHOLS ZENECA LIMITED (GB) 1994-12-08 WO disclosed