SCHEMBL5686703

SCHEMBL5686703

CCOC(C[C@H](CC(=O)OC(C)(C)C)NC(=O)[C@H](C)NC(=O)[C@@H](NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)C(C)O)C(C)CC)OCC

nearest known ligand 0.42

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
REN P00797 10/20 0.42
CTSB P07858 2/20 0.39
CTSK P43235 2/20 0.39
CTSD P07339 1/20 0.39
BACE1 P56817 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5686572 0.93 CASP1 (0.43) RENCTSBCTSKCTSDBACE1
SCHEMBL5686581 0.93 CASP1 (0.43) RENCTSBCTSKCTSDBACE1
SCHEMBL5686901 0.92 REN (0.46) RENCTSBCTSKCTSD
SCHEMBL5689425 0.87 CASP1 (0.49) RENCTSKCTSDBACE1
SCHEMBL7198017 0.86 REN (0.46) RENCTSBCTSKCTSD
SCHEMBL5686929 0.76 CASP1 (0.47) RENCTSBCTSKBACE1
SCHEMBL8026640 0.76 CASP1 (0.47) RENCTSBCTSKBACE1
SCHEMBL5686579 0.75 CTSD (0.38) CTSD
SCHEMBL5686711 0.74 CTSD (0.36) CTSDBACE1
SCHEMBL5686897 0.73 CTSD (0.37) CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0979241-B1 (3R)-3-AMINO-4-CARBOXYBUTYRALDEHYDE DERIVATIVES INHIBITING THE RELEASE OF INTERLEUKIN-1/BETA IVAX DRUG RES INST LTD (HU) 2006-03-01 EP disclosed
US-6593300-B1 Inhibitors of the interleukin-1 beta converting enzyme GYOGYSZERKUTATO INTEZET KFT. (HU) 2003-07-15 US disclosed