SCHEMBL5687616

SCHEMBL5687616

Nc1ccc(-c2cnccc2Br)c(O)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
TSHR P16473 1/20 0.37
CASP1 P29466 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
AXL P30530 1/20 0.36
EP300 Q09472 1/20 0.36
KAT2B Q92831 1/20 0.36
KAT8 Q9H7Z6 1/20 0.36
KDM4E B2RXH2 4/20 0.35
MAPT P10636 3/20 0.35
ALDH1A1 P00352 2/20 0.35
TDP1 Q9NUW8 2/20 0.35
IMPDH2 P12268 1/20 0.35
CYP3A4 P08684 1/20 0.34
GAA P10253 1/20 0.34
ESR2 Q92731 1/20 0.34
PTPN1 P18031 1/20 0.34
RPS6KA3 P51812 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5687575 0.79 TSHR (0.50) TSHRCASP1TDP1CYP3A4LCK
SCHEMBL5684611 0.79 CA1 (0.46) CA1CA2TSHRCASP1NPC1
SCHEMBL5685368 0.78 ALOX15 (0.54) CA1CA2TSHRRAB9AMAPT
SCHEMBL31064872 0.77 AXL (0.41) TSHRCASP1NPC1RAB9AAXL
SCHEMBL5684893 0.74 SMN1; SMN2 (0.45) CA1CA2TSHRCASP1NPC1
SCHEMBL29484239 0.74 CASP1 (0.59) CA1CA2TSHRCASP1NPC1
SCHEMBL483397 0.74 CASP1 (0.59) CA1CA2TSHRCASP1NPC1
Methane SCHEMBL28033104 0.72 CASP1 (0.56) CA1CA2TSHRCASP1NPC1
SCHEMBL5687682 0.72 IMPDH2 (0.50) CA1CA2TSHRCASP1NPC1
SCHEMBL5684882 0.71 AXL (0.59) NPC1RAB9AAXLKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7077872-B2 Oxidation hair dyes containing 3-aminophenol derivatives, and novel 3-aminophenol derivatives WELLA AG (DE) 2006-07-18 US disclosed
EP-1418879-B1 OXIDATION HAIR DYES CONTAINING 3-AMINOPHENOL DERIVATIVES, AND NOVEL 3-AMINOPHENOL DERIVATIVES WELLA AG (DE) 2006-04-12 EP disclosed
US-20040200010-A1 Oxidation hair dyes containing 3-aminophenol derivatives, and novel 3-aminophenol derivatives WELLA AKTIENGESELLSCHAFT (DE) 2004-10-14 US disclosed
EP-1418879-A1 OXIDATION HAIR DYES CONTAINING 3-AMINOPHENOL DERIVATIVES, AND NOVEL 3-AMINOPHENOL DERIVATIVES Wella Aktiengesellschaft (DE) 2004-05-19 EP disclosed
WO-2003017955-A1 OXIDATION HAIR DYES CONTAINING 3-AMINOPHENOL DERIVATIVES, AND NOVEL 3-AMINOPHENOL DERIVATIVES WELLA AKTIENGESELLSCHAFT (DE) 2003-03-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040200010-A1 Oxidation hair dyes containing 3-aminophenol derivatives, and novel 3-aminophenol derivatives KRT18, S100P, ALDH7A1 CA1 2105/4885CA2 675/4885TSHR 2675/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.