SCHEMBL568905

SCHEMBL568905

N#Cc1ccc(N)c(C(F)(F)F)c1

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 1/20 0.53
KIF11 P52732 2/20 0.47
AR P10275 4/20 0.40
GAA P10253 2/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
P4HB P07237 1/20 0.38
MRGPRX4 Q96LA9 1/20 0.38
SLC22A12 Q96S37 4/20 0.38
FFAR4 Q5NUL3 2/20 0.37
TMPRSS4 Q9NRS4 1/20 0.37
GLA P06280 1/20 0.36
POLB P06746 1/20 0.36
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4049024 0.85 KIF11 (0.63) TRPV4KIF11AR
SCHEMBL1724867 0.84 KIF11 (0.51) TRPV4KIF11ARGAAKDM4E
SCHEMBL29800340 0.83 FFAR4 (0.39) TRPV4KIF11ARGAAFFAR4
SCHEMBL7569957 0.81 TRPV4 (0.58) TRPV4KIF11ARP4HBMRGPRX4
SCHEMBL29353872 0.80 FFAR4 (0.37) TRPV4KIF11ARGAAFFAR4
SCHEMBL7116955 0.80 KIF11 (0.42) TRPV4KIF11GAAKDM4EALDH1A1
SCHEMBL20929103 0.80 FFAR4 (0.37) TRPV4KIF11ARGAAFFAR4
SCHEMBL7604551 0.79 TRPV4 (0.56) TRPV4KIF11ARGAAP4HB
SCHEMBL185191 0.78 KIF11 (0.58) TRPV4KIF11ARP4HBMRGPRX4
SCHEMBL10502974 0.78 TRPV4 (0.54) TRPV4KIF11ARP4HBMRGPRX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 136 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1301965-C Prepn process of 2-trifluoromethyl-4-cyano aniline DALIAN LUYUAN PHARMACEUTICAL I (CN) 2007-02-28 CN claimed
CN-1740147-A Prepn process of 2-trifluoromethyl-4-cyano aniline DALIAN LUYUAN PHARMACEUTICAL I (CN) 2006-03-01 CN claimed
JP-10204066-A None JP disclosed
US-20260090265-A1 COMPOUND, ORGANIC THIN FILM, PHOTOELECTRIC CONVERSION ELEMENT, IMAGE SENSOR, PHOTOSENSOR AND SOLID-STATE IMAGING APPARATUS MITSUBISHI GAS CHEMICAL COMPANY, INC. (JP) 2026-03-26 US disclosed
US-20250179072-A1 TRICYCLIC AKR1C3 DEPENDENT KARS INHIBITORS NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH, INC. 2025-06-05 US disclosed
CN-119930443-A Method for synthesizing trifluoromethyl substituted aniline by using tetradentate platinum complex as photocatalyst 九洲药业(杭州)有限公司 2025-05-06 CN disclosed
CN-114206870-B Tricyclic AKR1C 3-dependent KARS inhibitors 诺华股份有限公司 2024-09-03 CN disclosed
US-20240262827-A1 TRICYCLIC AKR1C3 DEPENDENT KARS INHIBITORS NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH, INC. 2024-08-08 US disclosed
WO-2024135508-A1 COMPOUND, ORGANIC THIN FILM, PHOTOELECTRIC CONVERSION ELEMENT, IMAGING ELEMENT, PHOTOSENSOR AND SOLID-STATE IMAGING DEVICE 三菱瓦斯化学株式会社 2024-06-27 WO disclosed
WO-2024126619-A1 ORGANIC ELECTROLUMINESCENT DEVICE COMPRISING A COMPOUND OF FORMULA (I) AND A COMPOUND OF FORMULA (II), AND DISPLAY DEVICE COMPRISING THE ORGANIC ELECTROLUMINESCENT DEVICE NOVALED GMBH (DE) 2024-06-20 WO disclosed
EP-4065117-B1 ISOQUINOLINE DERIVATIVES FOR USE IN TREATING GLUT1 DEFICIENCY SYNDROME GLIAPHARM SA (CH) 2024-06-19 EP disclosed
US-6362372-B2 HYDROGENATION OF A TRIFLUOROBENZYLNITRILE BY HYDROGEN IN AN ORGANIC SOLVENT IN THE PRESENCE OF AMMONIA AND A CATALYST COMPRISING A PLATINUM GROUP ELEMENT; EXTREMELY HIGH YIELDS CENTRAL GLASS COMPANY, LIMITED (JP) 2002-03-26 US disclosed
US-20020007086-A1 Process for producing trifluoromethylbenzylamines CENTRAL GLASS COMPANY, LIMITED (JP) 2002-01-17 US disclosed
US-6175041-B1 HYDROGENATING A TRIFLUOROMETHYLBENZONITRILE WITH HYDROGEN IN AN ORGANIC SOLVENT IN THE PRESENCE OF AMMONIA, USING A RANEY CATALYST CENTRAL GLASS COMPANY, LIMITED (JP) 2001-01-16 US disclosed
US-5981438-A HERBICIDE, INSECTICIDE AND PESTICIDE NIHON BAYER AGROCHEM K.K. (JP) 1999-11-09 US disclosed
CN-1194267-A 1-phenyl-5-anilinotetrazole compounds BAYER AGROCHEM KK (JP) 1998-09-30 CN disclosed
JP-H10204066-A 1-PHENYL-5-ANILINOTETRAZOLES AND THEIRS UTILIZATION AS AGROCHEMICAL NIPPON BAYER AGROCHEM KK 1998-08-04 JP disclosed
EP-0855394-A1 1-Phenyl-5-anilinotetrazoles derivatives, their preparation and their use as microbiocides, insecticides and/or herbicides NIHON BAYER AGROCHEM K.K. (JP) 1998-07-29 EP disclosed
US-4153687-A Derivatives, having an inhibitory action against protease and an antiphlogistic action, of the trypsin-kallikrein inhibitor obtained from cattle organs (BPTI), their preparation and their use as medicaments BAYER AKTIENGESELLSCHAFT (DE) 1979-05-08 US disclosed
US-4059402-A SUBLIMATION, MONOAZO DYES BAYER AKTIENGESELLSCHAFT (DT) 1977-11-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020007086-A1 Process for producing trifluoromethylbenzylamines IDH1, INMT, TH TRPV4 4031/4885KIF11 2157/4885AR 3622/4885
US-20250179072-A1 TRICYCLIC AKR1C3 DEPENDENT KARS INHIBITORS AKR1C2, AKR1B1, AKR1C1 TRPV4 3597/4885KIF11 571/4885AR 220/4885
US-20260090265-A1 COMPOUND, ORGANIC THIN FILM, PHOTOELECTRIC CONVERSION ELEMENT, IMAGE SENSOR, PHOTOSENSOR AND SOLID-STATE IMAGING APPARATUS SLC43A1, CNPY2, SCO2 TRPV4 508/4885KIF11 3758/4885AR 2057/4885
US-20240262827-A1 TRICYCLIC AKR1C3 DEPENDENT KARS INHIBITORS AKR1C2, AKR1B1, AKR1C1 TRPV4 3597/4885KIF11 571/4885AR 220/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.