SCHEMBL5692196

SCHEMBL5692196

CN(C)CCCN(CCCN(C)C)c1ccc(C#N)c(C(F)(F)F)c1.COCCN(C)c1ccc([N+](=O)[O-])cc1C(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGES O14684 1/20 0.38
AR P10275 14/20 0.37
PGR P06401 2/20 0.36
PIK3CD O00329 1/20 0.35
PIK3R1 P27986 1/20 0.35
PIK3CA P42336 1/20 0.35
PIK3CB P42338 1/20 0.35
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3058229 0.81 ALDH1A1 (0.45) ALDH1A1
SCHEMBL1408112 0.78 ALDH1A1 (0.46) PIK3CDPIK3R1PIK3CAPIK3CBALDH1A1
SCHEMBL3059882 0.78 AR (0.49) ARPGR
SCHEMBL1408560 0.73 ALDH1A1 (0.48) PIK3CDPIK3R1PIK3CBALDH1A1
SCHEMBL5693125 0.73 CYP3A4 (0.43) ARPGR
SCHEMBL5692286 0.72 VCAM1 (0.38) PGRPIK3CDPIK3R1PIK3CAPIK3CB
SCHEMBL2853583 0.72 VCAM1 (0.54) PTGESARALDH1A1
SCHEMBL3050476 0.71 AR (0.51) ARPGR
SCHEMBL5692157 0.71 MAPT (0.41) ARPGRALDH1A1
SCHEMBL3045088 0.69 AR (0.51) ARPGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1654221-A2 ANILINE DERIVATIVED ANDROGEN-, GLUCOCORTICOID-, MINERALCORTICOID- AND PROGESTERONE- RECEPTOR MODULATORS SMITHKLINE BEECHAM CORPORATION (US) 2006-05-10 EP disclosed
WO-2005000795-A2 ANILINE DERIVATIVED ANDROGEN-, GLUCOCORTICOID-, MINERALCORTICOID- AND PROGESTERONE- RECEPTOR MODULATORS SMITHKLINE BEECHAM CORPORATION (US) 2005-01-06 WO disclosed