SCHEMBL5693121

SCHEMBL5693121

CCCCN(C)c1ccc([N+](=O)[O-])cc1Cl.CCCCN(CCC)c1ccc(C#N)c(Cl)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.46
VCAM1 P19320 2/20 0.40
PGR P06401 4/20 0.39
LMNA P02545 2/20 0.36
HTT P42858 2/20 0.36
ALDH1A1 P00352 2/20 0.35
GAA P10253 1/20 0.35
CYP19A1 P11511 2/20 0.34
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
MCL1 Q07820 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
RECQL P46063 1/20 0.33
HCAR3 P49019 1/20 0.33
TP53 P04637 1/20 0.32
PIK3CD O00329 1/20 0.32
PIK3R1 P27986 1/20 0.32
PIK3CA P42336 1/20 0.32
PIK3CB P42338 1/20 0.32
HSD17B10 Q99714 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5692155 0.92 MAPT (0.46) MAPTVCAM1PGRLMNAHTT
SCHEMBL3060338 0.81 MAPT (0.60) MAPTVCAM1LMNAHTTALDH1A1
SCHEMBL3060094 0.80 PGR (0.54) PGR
SCHEMBL3054008 0.78 PGR (0.56) PGR
SCHEMBL6819352 0.77 MAPT (0.54) MAPTVCAM1LMNAHTTALDH1A1
SCHEMBL5692532 0.76 PGR (0.43) MAPTVCAM1PGRALDH1A1CYP19A1
SCHEMBL3060099 0.75 PGR (0.54) PGR
SCHEMBL3057818 0.75 VCAM1 (0.47) MAPTVCAM1ALDH1A1CYP19A1HCAR3
SCHEMBL5692492 0.74 MAPT (0.42) MAPTVCAM1PGRLMNAHTT
SCHEMBL5693113 0.74 MAPT (0.39) MAPTVCAM1PGRLMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1654221-A2 ANILINE DERIVATIVED ANDROGEN-, GLUCOCORTICOID-, MINERALCORTICOID- AND PROGESTERONE- RECEPTOR MODULATORS SMITHKLINE BEECHAM CORPORATION (US) 2006-05-10 EP disclosed
WO-2005000795-A2 ANILINE DERIVATIVED ANDROGEN-, GLUCOCORTICOID-, MINERALCORTICOID- AND PROGESTERONE- RECEPTOR MODULATORS SMITHKLINE BEECHAM CORPORATION (US) 2005-01-06 WO disclosed