SCHEMBL5696261

SCHEMBL5696261

CC(C)CCOc1ccc(C(C)C(=O)O)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.66
GAA P10253 1/20 0.65
HTT P42858 1/20 0.65
EPHX2 P34913 1/20 0.58
TP53 P04637 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
TDP1 Q9NUW8 1/20 0.54
TSHR P16473 2/20 0.53
ALDH1A1 P00352 1/20 0.53
THRB P10828 1/20 0.53
HSD17B10 Q99714 1/20 0.53
PTGS2 P35354 5/20 0.53
PTGS1 P23219 4/20 0.53
AKR1C3 P42330 4/20 0.53
AKR1C2 P52895 3/20 0.53
LMNA P02545 2/20 0.53
CYP2C9 P11712 2/20 0.53
CXCR1 P25024 2/20 0.53
CXCR2 P25025 2/20 0.53
RARB P10826 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7403967 0.85 GPR88 (0.59) PTGS2PTGS1AKR1C3AKR1C2LMNA
SCHEMBL8403335 0.85 GPR88 (0.59) PTGS2PTGS1AKR1C3AKR1C2LMNA
SCHEMBL14599721 0.85 GPR88 (0.59) MAPK1TP53SMN1; SMN2TSHRPTGS2
SCHEMBL1346573 0.83 POLB (0.51) GAAHTTTDP1TSHRPTGS2
SCHEMBL8463046 0.83 AKR1C3 (0.51) MAPK1GAAHTTTDP1TSHR
SCHEMBL11595380 0.83 POLB (0.51) GAAHTTTDP1TSHRPTGS2
SCHEMBL1749031 0.83 MAPT (0.60) TSHRPTGS2PTGS1AKR1C3AKR1C2
SCHEMBL9861070 0.82 LMNA (0.62) TP53TDP1TSHRAKR1C3AKR1C2
SCHEMBL11597542 0.82 PPARG (0.51) GAAHTTTDP1TSHRALDH1A1
SCHEMBL5881684 0.81 AKR1C3 (0.73) TSHRALDH1A1PTGS2PTGS1AKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1654218-A2 MATRIX METALLOPROTEINASE INHIBITORS GLAXO GROUP LIMITED (GB) 2006-05-10 EP disclosed
WO-2005016868-A2 MATRIX METALLOPROTEINASE INHIBITORS GLAXO GROUP LIMITED (GB) 2005-02-24 WO disclosed