SCHEMBL5698458

SCHEMBL5698458

C[S+]([O-])c1ccc(C2=C(c3ccc(C(F)(F)F)cc3)CCC2)cc1

nearest known ligand 0.59

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 10/20 0.59
PTGS1 P23219 4/20 0.55
MAPK14 Q16539 1/20 0.38
KIF11 P52732 6/20 0.36
CYP1A2 P05177 1/20 0.34
OPRM1 P35372 1/20 0.34
OPRL1 P41146 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4362915 0.82 OPRM1 (0.40) KIF11OPRM1OPRL1
SCHEMBL16622528 0.82 OPRM1 (0.40) KIF11OPRM1OPRL1
SCHEMBL6687073 0.81 PTGS2 (0.56) PTGS2PTGS1MAPK14
SCHEMBL5698516 0.80 PTGS2 (0.54) PTGS2PTGS1MAPK14
SCHEMBL5698535 0.75 PTGS2 (0.58) PTGS2PTGS1
SCHEMBL8993560 0.75 PTGS2 (0.34) PTGS2PTGS1MAPK14
SCHEMBL215443 0.74 PTGS2 (1.00) PTGS2PTGS1
SCHEMBL8654658 0.73 PTGS2 (0.58) PTGS2PTGS1MAPK14KIF11CYP1A2
SCHEMBL8371975 0.72 PTGS2 (0.44) PTGS2PTGS1
SCHEMBL8651596 0.71 PTGS2 (1.00) PTGS2PTGS1KIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1682143-A2 COMBINATIONS COMPRISING AN HSP90 INHIBITOR AND A PHOPHODIESTERASE INHIBITOR FOR TREATING OR PREVENTING NEOPLASIA Pharmacia Corporation (US) 2006-07-26 EP disclosed
WO-2005041879-A2 COMBINATIONS COMPRISING AN Hsp90 INHIBITOR AND A PHOPHODIESTERASE INHIBITOR FOR TREATING OR PREVENTING NEOPLASIA PHARMACIA CORPORATION (US) 2005-05-12 WO disclosed
EP-1283723-A2 COMBINATION THERAPY USING COX-2 SELECTIVE INHIBITOR AND THROMBOXANE INHIBITOR AND COMPOSITIONS THEREFOR Merck Frosst Canada & Co. (CA) 2003-02-19 EP disclosed
WO-2001087343-A2 COMBINATION THERAPY USING COX-2 SELECTIVE INHIBITOR AND THROMBOXANE INHIBITOR AND COMPOSITIONS THEREFOR MERCK FROSST CANADA & CO. (CA) 2001-11-22 WO disclosed