SCHEMBL5699092

SCHEMBL5699092

CONc1ncnc2nc[nH]c12

nearest known ligand 0.60

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTT P42858 6/20 0.60
LMNA P02545 5/20 0.60
PDPK1 O15530 1/20 0.56
CYP1A2 P05177 2/20 0.55
PAK1 Q13153 1/20 0.55
HIF1A Q16665 1/20 0.55
HSD17B10 Q99714 2/20 0.54
PKM P14618 1/20 0.54
SMN1; SMN2 Q16637 3/20 0.54
LCK P06239 1/20 0.54
MAPT P10636 1/20 0.54
CYP3A4 P08684 1/20 0.53
NPC1 O15118 2/20 0.52
RAB9A P51151 2/20 0.52
MKNK1 Q9BUB5 1/20 0.52
CDK2 P24941 1/20 0.51
BRD4 O60885 3/20 0.51
TP53 P04637 1/20 0.51
TSHR P16473 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fluoride SCHEMBL31379723 0.98 HTT (0.59) HTTLMNAPDPK1CYP1A2PAK1
SCHEMBL21914 0.79 HTT (0.62) HTTLMNACYP1A2PAK1HIF1A
SCHEMBL29380490 0.79 HTT (0.62) HTTLMNACYP1A2PAK1HIF1A
SCHEMBL10918760 0.78 HTT (0.60) HTTLMNAPDPK1CYP1A2PAK1
SCHEMBL6243538 0.78 HTT (0.60) HTTLMNAPDPK1CYP1A2PAK1
SCHEMBL11591794 0.77 HTT (0.59) HTTLMNACYP1A2PAK1HIF1A
SCHEMBL405823 0.76 HTT (0.58) HTTLMNACYP1A2PAK1HIF1A
SCHEMBL6509992 0.76 XDH (0.45) HTTLMNAMAPT
SCHEMBL29501839 0.76 LMNA (0.57) HTTLMNACYP1A2PAK1HSD17B10
SCHEMBL17901710 0.76 HTT (0.57) HTTLMNACYP1A2PAK1HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 54 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025013869-A1 FLUORINE-CONTAINING POLYMER HAVING NITROGEN-CONTAINING AROMATIC RING, PRODUCTION METHOD THEREFOR, AND COMPOSITION THEREOF ダイキン工業株式会社 2025-01-16 WO claimed
US-20060223148-A1 Process for sequence saturation mutagenesis (sesam) BASF AKTIENGESCHAFT (DE) 2006-10-05 US claimed
WO-1998001459-A1 NOVEL N-ALKOXYADENINE DERIVATIVES ACTING AS CYTOKINE INHIBITORS NOVO NORDISK A/S (DK) 1998-01-15 WO claimed
US-12492428-B2 Methods and compositions for the quantitation of mitochondrial nucleic acid AGENA BIOSCIENCE, INC. (US) 2025-12-09 US disclosed
US-12473595-B2 Coupling method OXFORD NANOPORE TECHNOLOGIES PLC (GB) 2025-11-18 US disclosed
US-20250290132-A1 COUPLING METHOD OXFORD NANOPORE TECHNOLOGIES PLC (GB) 2025-09-18 US disclosed
EP-4574993-A2 METHODS AND PROCESSES FOR NON-INVASIVE ASSESSMENT OF GENETIC VARIATIONS Sequenom, Inc. (US) 2025-06-25 EP disclosed
US-20250157582-A1 METHODS AND PROCESSES FOR NON-INVASIVE ASSESSMENT OF GENETIC VARIATIONS SEQUENOM, INC. 2025-05-15 US disclosed
EP-3540076-B1 METHODS AND PROCESSES FOR NON-INVASIVE ASSESSMENT OF GENETIC VARIATIONS SEQUENOM INC (US) 2025-05-07 EP disclosed
WO-2025013869-A1 FLUORINE-CONTAINING POLYMER HAVING NITROGEN-CONTAINING AROMATIC RING, PRODUCTION METHOD THEREFOR, AND COMPOSITION THEREOF ダイキン工業株式会社 2025-01-16 WO disclosed
CN-118119404-A Immunogenic LNP compositions and methods thereof 辉瑞公司 2024-05-31 CN disclosed
EP-1307592-A2 SINGLE-LABELED OLIGONUCLEOTIDE PROBES University of Utah Research Foundation (US) 2003-05-07 EP disclosed
US-20030022177-A1 Single-labeled oligonucleotide probes for homogeneous nucleic acid sequence analysis NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2003-01-30 US disclosed
WO-2002085309-A2 COMPOSITION, FORMULATIONS & KITS FOR TREATMENT OF RESPIRATORY & LUNG DISEASE WITH ANTI-SENSE OLIGONUCLEOTIDES & A BRONCHODILATING AGENT EPIGENESIS PHARMACEUTICALS, INC. (US) 2002-10-31 WO disclosed
WO-2002014555-A2 SINGLE-LABELED OLIGONUCLEOTIDE PROBES UNIVERSITY OF UTAH RESEARCH FOUNDATION (US) 2002-02-21 WO disclosed
EP-1168919-A2 LOW ADENOSINE ANTI-SENSE OLIGONUCLEOTIDE, COMPOSITIONS, KIT AND METHOD FOR TREATMENT OF AIRWAY DISORDERS ASSOCIATED WITH BRONCHOCONSTRICTION, LUNG INFLAMMATION, ALLERGY(IES) AND SURFACTANT DEPLETION East Carolina University (US) 2002-01-09 EP disclosed
WO-2000062736-A2 LOW ADENOSINE ANTI-SENSE OLIGONUCLEOTIDE, COMPOSITIONS, KIT AND METHOD FOR TREATMENT OF AIRWAY DISORDERS ASSOCIATED WITH BRONCHOCONSTRICTION, LUNG INFLAMMATION, ALLERGY(IES) AND SURFACTANT DEPLETION EAST CAROLINA UNIVERSITY (US) 2000-10-26 WO disclosed
EP-0973788-A1 TRICYCLIC BASE ANALOGUES Amersham Pharmacia Biotech UK Limited (GB) 2000-01-26 EP disclosed
WO-1998043991-A1 TRICYCLIC BASE ANALOGUES AMERSHAM PHARMACIA BIOTECH UK LIMITED (GB) 1998-10-08 WO disclosed
WO-1998001459-A1 NOVEL N-ALKOXYADENINE DERIVATIVES ACTING AS CYTOKINE INHIBITORS NOVO NORDISK A/S (DK) 1998-01-15 WO disclosed