SCHEMBL5699201

SCHEMBL5699201

CCOC(=O)c1[nH]c2ccc(N)c(Cc3ccccc3)c2c1-c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.54
HPGD P15428 4/20 0.54
CYP1A2 P05177 1/20 0.54
XBP1 P17861 1/20 0.54
CYP2C19 P33261 1/20 0.54
PDE3B Q13370 1/20 0.46
PDE3A Q14432 1/20 0.46
TP53 P04637 3/20 0.45
HTR6 P50406 1/20 0.44
CSF1R P07333 1/20 0.43
MAPT P10636 7/20 0.43
NPC1 O15118 4/20 0.43
RAB9A P51151 4/20 0.43
KDM4E B2RXH2 3/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
GAA P10253 2/20 0.43
TDP1 Q9NUW8 1/20 0.43
GRM6 O15303 1/20 0.42
MDM2 Q00987 1/20 0.42
KMT2A Q03164 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5738434 0.80 ALDH1A1 (0.56) ALDH1A1HPGDCYP1A2XBP1CYP2C19
SCHEMBL11300000 0.78 ALDH1A1 (0.65) ALDH1A1HPGDCYP1A2XBP1CYP2C19
SCHEMBL5737293 0.75 ALDH1A1 (0.46) ALDH1A1HPGDCYP1A2XBP1CYP2C19
SCHEMBL5206974 0.74 ALDH1A1 (0.54) ALDH1A1HPGDCYP1A2XBP1CYP2C19
SCHEMBL6346608 0.73 RAB9A (0.55) ALDH1A1PDE3BPDE3ATP53MAPT
SCHEMBL7671532 0.73 HTR6 (0.68) ALDH1A1HPGDTP53HTR6MAPT
SCHEMBL5738353 0.73 ALDH1A1 (0.42) ALDH1A1HPGDCYP1A2XBP1CYP2C19
SCHEMBL2956667 0.73 ALDH1A1 (0.73) ALDH1A1HPGDCYP1A2XBP1CYP2C19
SCHEMBL5204639 0.73 ALDH1A1 (0.53) ALDH1A1HPGDCYP1A2XBP1CYP2C19
SCHEMBL8538896 0.72 ALDH1A1 (0.50) ALDH1A1HPGDCYP1A2XBP1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1682530-A1 SUBSTITUTED PYRROLE-INDOLES AS INHIBITORS OF PAI-1 Wyeth (US) 2006-07-26 EP disclosed
WO-2005030756-A1 SUBSTITUTED PYRROLE-INDOLES AS INHIBITORS OF PAI-1 WYETH (US) 2005-04-07 WO disclosed