SCHEMBL5700847

SCHEMBL5700847

COC(=O)CC(NC(=O)c1ccc(OC)c(OC)c1)c1ccc(N)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 4/20 0.54
ROCK1 Q13464 4/20 0.54
TAS1R3 Q7RTX0 2/20 0.51
TAS1R1 Q7RTX1 2/20 0.51
TNF P01375 3/20 0.49
LMNA P02545 2/20 0.48
MAPT P10636 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
HPGD P15428 1/20 0.46
ALDH1A1 P00352 1/20 0.46
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
PDE4A P27815 2/20 0.44
PDE4B Q07343 2/20 0.44
PDE4C Q08493 2/20 0.44
PDE4D Q08499 2/20 0.44
ANPEP P15144 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
FLT3 P36888 1/20 0.43
NR1H4 Q96RI1 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5700841 1.00 ROCK2 (0.54) ROCK2ROCK1TAS1R3TAS1R1TNF
SCHEMBL7876199 0.93 HPGD (0.52) ROCK2ROCK1TAS1R3TAS1R1TNF
SCHEMBL7867559 0.85 ITGB3 (0.49) ROCK2ROCK1TAS1R3TAS1R1TNF
SCHEMBL5700999 0.83 MAPT (0.49) ROCK2ROCK1LMNAMAPTALDH1A1
SCHEMBL5701002 0.83 MAPT (0.49) ROCK2ROCK1LMNAMAPTALDH1A1
SCHEMBL5700932 0.81 MEN1 (0.60) ROCK2ROCK1LMNAMAPTMEN1
SCHEMBL5700925 0.81 MEN1 (0.60) ROCK2ROCK1LMNAMAPTMEN1
SCHEMBL7876448 0.81 POLB (0.58) ROCK2ROCK1TAS1R3TAS1R1TNF
SCHEMBL7872607 0.80 TAS1R3 (0.53) ROCK2ROCK1TAS1R3TAS1R1TNF
SCHEMBL15595838 0.78 TAS1R3 (0.55) TAS1R3TAS1R1LMNAMAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1027328-B1 SUBSTITUTED ANILIDES AVENTIS PHARMA LTD (GB) 2006-08-23 EP disclosed
US-6479519-B1 INHIBITORS OF CELL ADHESION; TREATMENT OF ASTHMA OR INFLAMMATORY BOWEL DISEASE AVENTIS PHARMA LIMITED (GB) 2002-11-12 US disclosed