SCHEMBL5704149

SCHEMBL5704149

CS(=O)(=O)NC(=O)c1ccc(OBOc2ccc(C(=O)NS(C)(=O)=O)c(OCCF)c2)cc1OCCF

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 16/20 0.43
SCN5A Q14524 1/20 0.41
GRM2 Q14416 1/20 0.40
ADRB1 P08588 1/20 0.38
ADRB3 P13945 1/20 0.38
ALDH1A1 P00352 1/20 0.37
TP53 P04637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5703853 0.86 KDM4E (0.46) SCN9ASCN5AGRM2ADRB1ADRB3
SCHEMBL4582967 0.81 SCN9A (0.43) SCN9ASCN5AGRM2ADRB1ADRB3
SCHEMBL5703690 0.80 ADRB3 (0.46) SCN9AADRB1ADRB3ALDH1A1TP53
SCHEMBL5703997 0.75 SCN9A (0.55) SCN9AADRB1ADRB3
SCHEMBL22444820 0.70 CXCR2 (0.50) SCN9AADRB1ADRB3ALDH1A1TP53
SCHEMBL22067283 0.69 KCNMA1 (0.48) SCN9AADRB1ADRB3
SCHEMBL7991086 0.69 ALDH1A1 (0.56) GRM2ADRB1ADRB3ALDH1A1TP53
SCHEMBL4585857 0.68 KDM4E (0.44) SCN9AADRB1ADRB3
SCHEMBL4584315 0.66 ADRB1 (0.42) SCN9ASCN5AGRM2ADRB1ADRB3
SCHEMBL16319476 0.65 SCN9A (0.59) SCN9ASCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1697301-A2 AMINOALCOHOL DERIVATIVES Astellas Pharma Inc. (JP) 2006-09-06 EP disclosed
WO-2005061433-A2 AMINOALCOHOL DERIVATIVES ASTELLAS PHARMA INC. (JP) 2005-07-07 WO disclosed