SCHEMBL5705461

SCHEMBL5705461

CC(O)c1ncnc(NCCc2ccc(OC(F)(F)F)cc2)c1I

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VNN1 O95497 2/20 0.39
TP53 P04637 1/20 0.38
ABL1 P00519 2/20 0.37
BCR P11274 2/20 0.37
CASR P41180 1/20 0.37
AURKA O14965 1/20 0.37
RPS6KB1 P23443 1/20 0.37
CYP3A4 P08684 2/20 0.37
ACACB O00763 1/20 0.36
LTA4H P09960 1/20 0.36
EPHX2 P34913 1/20 0.36
CNR2 P34972 2/20 0.36
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
FAAH O00519 3/20 0.35
RAB9A P51151 1/20 0.35
GALR3 O60755 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5705467 0.91 TP53 (0.39) VNN1TP53ABL1BCRAURKA
SCHEMBL5705458 0.89 CYP3A4 (0.39) VNN1TP53ABL1BCRAURKA
SCHEMBL5705522 0.89 TP53 (0.38) VNN1TP53ABL1BCRAURKA
SCHEMBL5705471 0.86 VNN1 (0.40) VNN1TP53ABL1BCRAURKA
SCHEMBL5705416 0.81 MAPK1 (0.50) ACACBCNR2MAPTRAB9AHTT
Flufenerim SCHEMBL29429245 0.80 CYP3A4 (0.42) TP53ABL1BCRCYP3A4CNR2
Flufenerim SCHEMBL26581 0.80 CYP3A4 (0.42) TP53ABL1BCRCYP3A4CNR2
SCHEMBL27993030 0.76 CYP3A4 (0.39) VNN1TP53ABL1BCRCYP3A4
SCHEMBL9038247 0.75 HTT (0.39) TP53AURKARPS6KB1CNR2POLB
SCHEMBL5705465 0.74 HTR7 (0.46) TP53POLBMAPTRAB9AGALR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1074546-B1 5-IODO-4-PHENETHYLAMINOPYRIMIDINE DERIVATIVES, INTERMEDIATES THEREOF, PROCESS FOR PRODUCING THE SAME AND AGRICULTURAL/HORTICULTURAL PESTICIDES UBE INDUSTRIES (JP) 2006-09-06 EP claimed
US-6521627-B1 Insecticidal, acaricidal, nematocidal and fungicidal activities UBE INDUSTRIES, LTD. (JP) 2003-02-18 US claimed
EP-1074546-A1 5-IODO-4-PHENETHYLAMINOPYRIMIDINE DERIVATIVES, INTERMEDIATES THEREOF, PROCESS FOR PRODUCING THE SAME AND AGRICULTURAL/HORTICULTURAL PESTICIDES Ube Industries, Ltd. (JP) 2001-02-07 EP claimed
EP-1074546-B1 5-IODO-4-PHENETHYLAMINOPYRIMIDINE DERIVATIVES, INTERMEDIATES THEREOF, PROCESS FOR PRODUCING THE SAME AND AGRICULTURAL/HORTICULTURAL PESTICIDES UBE INDUSTRIES (JP) 2006-09-06 EP disclosed
US-6521627-B1 Insecticidal, acaricidal, nematocidal and fungicidal activities UBE INDUSTRIES, LTD. (JP) 2003-02-18 US disclosed
EP-1074546-A1 5-IODO-4-PHENETHYLAMINOPYRIMIDINE DERIVATIVES, INTERMEDIATES THEREOF, PROCESS FOR PRODUCING THE SAME AND AGRICULTURAL/HORTICULTURAL PESTICIDES Ube Industries, Ltd. (JP) 2001-02-07 EP disclosed