SCHEMBL5705471

SCHEMBL5705471

CC(=O)OC(C)c1ncnc(NCCc2ccc(OC(F)(F)F)cc2)c1I

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VNN1 O95497 3/20 0.40
AURKA O14965 1/20 0.38
RPS6KB1 P23443 1/20 0.38
ACACB O00763 1/20 0.37
LTA4H P09960 1/20 0.37
EPHX2 P34913 1/20 0.37
CYP3A4 P08684 1/20 0.35
HTT P42858 1/20 0.35
TRPV1 Q8NER1 2/20 0.35
EPHX1 P07099 1/20 0.35
ALOX5 P09917 1/20 0.35
PPARG P37231 1/20 0.35
TP53 P04637 1/20 0.34
ABL1 P00519 2/20 0.34
BCR P11274 2/20 0.34
CYP2C9 P11712 1/20 0.34
P2RX3 P56373 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HDAC3 O15379 1/20 0.34
HDAC4 P56524 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5705461 0.86 VNN1 (0.39) VNN1AURKARPS6KB1ACACBLTA4H
SCHEMBL5705467 0.86 TP53 (0.39) VNN1AURKARPS6KB1LTA4HEPHX2
SCHEMBL5705455 0.85 MAPK1 (0.43) AURKAACACBHTTHDAC3HDAC1
SCHEMBL5705522 0.84 TP53 (0.38) VNN1AURKARPS6KB1LTA4HEPHX2
SCHEMBL5705458 0.84 CYP3A4 (0.39) VNN1AURKARPS6KB1LTA4HEPHX2
SCHEMBL9038563 0.78 HTT (0.40) AURKARPS6KB1ACACBHTTTP53
Flufenerim SCHEMBL26581 0.75 CYP3A4 (0.42) CYP3A4HTTTRPV1TP53ABL1
Flufenerim SCHEMBL29429245 0.75 CYP3A4 (0.42) CYP3A4HTTTRPV1TP53ABL1
SCHEMBL9038157 0.74 GALR3 (0.50) AURKARPS6KB1HTTTP53
SCHEMBL27993030 0.71 CYP3A4 (0.39) VNN1LTA4HEPHX2CYP3A4HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1074546-B1 5-IODO-4-PHENETHYLAMINOPYRIMIDINE DERIVATIVES, INTERMEDIATES THEREOF, PROCESS FOR PRODUCING THE SAME AND AGRICULTURAL/HORTICULTURAL PESTICIDES UBE INDUSTRIES (JP) 2006-09-06 EP claimed
US-6521627-B1 Insecticidal, acaricidal, nematocidal and fungicidal activities UBE INDUSTRIES, LTD. (JP) 2003-02-18 US claimed
EP-1074546-A1 5-IODO-4-PHENETHYLAMINOPYRIMIDINE DERIVATIVES, INTERMEDIATES THEREOF, PROCESS FOR PRODUCING THE SAME AND AGRICULTURAL/HORTICULTURAL PESTICIDES Ube Industries, Ltd. (JP) 2001-02-07 EP claimed
EP-1074546-B1 5-IODO-4-PHENETHYLAMINOPYRIMIDINE DERIVATIVES, INTERMEDIATES THEREOF, PROCESS FOR PRODUCING THE SAME AND AGRICULTURAL/HORTICULTURAL PESTICIDES UBE INDUSTRIES (JP) 2006-09-06 EP disclosed
US-6521627-B1 Insecticidal, acaricidal, nematocidal and fungicidal activities UBE INDUSTRIES, LTD. (JP) 2003-02-18 US disclosed
EP-1074546-A1 5-IODO-4-PHENETHYLAMINOPYRIMIDINE DERIVATIVES, INTERMEDIATES THEREOF, PROCESS FOR PRODUCING THE SAME AND AGRICULTURAL/HORTICULTURAL PESTICIDES Ube Industries, Ltd. (JP) 2001-02-07 EP disclosed