SCHEMBL5706202

SCHEMBL5706202

CN(c1ccc(Br)cc1)C1CCCCCC1.[MgH2]

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
TRPV1 Q8NER1 1/20 0.38
HRH4 Q9H3N8 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37
ABCB11 O95342 1/20 0.36
ADORA3 P0DMS8 1/20 0.36
AR P10275 1/20 0.36
CYP2D6 P10635 1/20 0.36
SLC6A2 P23975 1/20 0.36
PDE4A P27815 1/20 0.36
SLC6A4 P31645 1/20 0.36
SLC6A3 Q01959 1/20 0.36
KCNH2 Q12809 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
LMNA P02545 3/20 0.36
NPSR1 Q6W5P4 1/20 0.36
GAA P10253 1/20 0.36
JAK3 P52333 5/20 0.36
JAK1 P23458 4/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4173780 1.00 MEN1 (0.42) MEN1KMT2ATRPV1HRH4HRH3
SCHEMBL4168246 0.98 MEN1 (0.43) MEN1KMT2ATRPV1HRH4HRH3
Methylamine SCHEMBL28816853 0.94 MEN1 (0.41) MEN1KMT2ATRPV1HRH4HRH3
Methylamine SCHEMBL28000605 0.93 MEN1 (0.40) MEN1KMT2ATRPV1HRH4HRH3
SCHEMBL3717754 0.88 CYP2A6 (0.36) MEN1KMT2AHRH3SLC6A4HTT
SCHEMBL4485887 0.88 HRH4 (0.44) MEN1KMT2ATRPV1HRH4HRH3
SCHEMBL7793337 0.80 ALDH1A1 (0.44) MEN1KMT2ATRPV1HRH4HRH3
SCHEMBL25353462 0.79 KDM1A (0.38) MEN1KMT2AKCNH2LMNAHTT
SCHEMBL26011715 0.79 NMT1 (0.35) SLC6A2SLC6A4SLC6A3
SCHEMBL15013072 0.78 TRPA1 (0.49) TRPV1HRH4HRH3KCNH2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1219632-B1 STEROIDS, THEIR PREPARATION, PHARMACEUTICAL COMPOSITIONS THEREOF AND USES OF THE COMPOUNDS SHANGHAI ZHONGXI PHARMACEUTICA (CN) 2006-10-25 EP disclosed
US-6514956-B1 For treating diseases associated with progestogen dependence and for fertility control, abortion or contraception and for anticancer use SHANGHAI ZHONGXI PHARMACEUTICAL CO., LTD. (CN) 2003-02-04 US disclosed
EP-1219632-A1 STEROIDS, THEIR PREPARATION, PHARMACEUTICAL COMPOSITIONS THEREOF AND USES OF THE COMPOUNDS Shanghai Zhongxi Pharmaceutical Co. Ltd. (CN) 2002-07-03 EP disclosed