SCHEMBL5707683

SCHEMBL5707683

O=C1C(=O)N(c2ccc([N+](=O)[O-])cc2)c2ccccc21

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN2A Q99250 2/20 0.69
ALDH1A1 P00352 3/20 0.65
GAA P10253 3/20 0.65
BCHE P06276 2/20 0.65
CES1 P23141 2/20 0.65
CES2 O00748 1/20 0.65
NPSR1 Q6W5P4 1/20 0.65
HPGD P15428 1/20 0.49
HTT P42858 1/20 0.49
IDO1 P14902 1/20 0.47
TDO2 P48775 1/20 0.47
TTR P02766 1/20 0.47
PTPRC P08575 2/20 0.45
ACHE P22303 2/20 0.45
S100A4 P26447 1/20 0.45
CA12 O43570 2/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA9 Q16790 1/20 0.45
CASP1 P29466 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9330406 0.84 SCN2A (0.71) SCN2AALDH1A1GAABCHECES1
SCHEMBL9330569 0.82 CASP1 (0.61) SCN2AALDH1A1GAABCHECES1
SCHEMBL30118348 0.82 SCN2A (1.00) SCN2AALDH1A1GAAIDO1TDO2
SCHEMBL1973251 0.82 SCN2A (1.00) SCN2AALDH1A1GAAIDO1TDO2
Phenyl Isatin SCHEMBL916808 0.79 CES1 (1.00) ALDH1A1GAABCHECES1CES2
SCHEMBL5707675 0.79 MEN1 (0.48) SCN2AALDH1A1GAABCHECES1
SCHEMBL10399763 0.78 SCN2A (0.56) SCN2AALDH1A1GAAHTTTTR
SCHEMBL10399765 0.78 SCN2A (0.56) SCN2AALDH1A1GAAHTTTTR
SCHEMBL5707613 0.78 ALDH1A1 (0.54) ALDH1A1GAABCHECES1CES2
SCHEMBL14830299 0.77 CES1 (0.73) ALDH1A1GAABCHECES1CES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1705227-A2 New dyestuffs and colorants with specific carbonyl compounds Henkel Kommanditgesellschaft auf Aktien (DE) 2006-09-27 EP claimed
EP-1705227-A2 New dyestuffs and colorants with specific carbonyl compounds Henkel Kommanditgesellschaft auf Aktien (DE) 2006-09-27 EP disclosed
EP-0369344-B1 N-arylation of isatins ABBOTT LAB (US) 1994-04-06 EP disclosed
US-5151518-A N-arylation of isatins ABBOTT LABORATORIES (US) 1992-09-29 US disclosed
EP-0369344-A1 N-arylation of isatins ABBOTT LABORATORIES (US) 1990-05-23 EP disclosed