SCHEMBL5712342

SCHEMBL5712342

CCCCOc1c(Cl)cc(C=O)cc1OC.O=Cc1cc(O)c(O)c(Cl)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.46
L3MBTL1 Q9Y468 3/20 0.46
HTT P42858 4/20 0.43
S1PR2 O95136 1/20 0.43
S1PR1 P21453 1/20 0.43
S1PR3 Q99500 1/20 0.43
LPAR2 Q9HBW0 1/20 0.43
KMT2A Q03164 4/20 0.42
MAPT P10636 5/20 0.42
MEN1 O00255 3/20 0.42
HPGD P15428 3/20 0.42
LMNA P02545 1/20 0.42
GAA P10253 1/20 0.42
ALPG P10696 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
HSD17B10 Q99714 1/20 0.41
TDP1 Q9NUW8 3/20 0.41
POLB P06746 3/20 0.41
MAPK1 P28482 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4007449 0.90 ALDH1A1 (0.51) ALDH1A1L3MBTL1HTTS1PR2S1PR1
SCHEMBL14195847 0.85 S1PR2 (0.53) ALDH1A1L3MBTL1HTTS1PR2S1PR1
SCHEMBL13221149 0.83 ALDH1A1 (0.53) ALDH1A1L3MBTL1HTTS1PR2S1PR1
SCHEMBL4005149 0.83 ALDH1A1 (0.46) ALDH1A1L3MBTL1HTTS1PR2S1PR1
SCHEMBL7462928 0.80 FDPS (0.51) ALDH1A1HTTKMT2AMAPTMEN1
SCHEMBL14195840 0.80 ALDH1A1 (0.45) ALDH1A1HPGDTDP1MAPK1ALOX5
SCHEMBL15771884 0.79 ALDH1A1 (0.51) ALDH1A1L3MBTL1HTTKMT2AMAPT
SCHEMBL5712326 0.79 S1PR2 (0.46) ALDH1A1L3MBTL1HTTS1PR2S1PR1
SCHEMBL18033266 0.77 FDPS (0.45) ALDH1A1HTTKMT2AMAPTMEN1
SCHEMBL2650454 0.77 ALDH1A1 (0.48) ALDH1A1L3MBTL1HTTKMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1383736-A4 PEPTIDE DEFORMYLASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2006-04-19 EP disclosed
EP-1383736-A2 PEPTIDE DEFORMYLASE INHIBITORS SmithKline Beecham Corporation (US) 2004-01-28 EP disclosed
WO-2003002522-A1 PEPTIDE DEFORMYLASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2003-01-09 WO disclosed