SCHEMBL5712945

SCHEMBL5712945

Cc1cc([N+](=O)[O-])ccc1[C]=O

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.62
TSHR P16473 5/20 0.62
TDP1 Q9NUW8 4/20 0.62
CYP3A4 P08684 4/20 0.58
ACHE P22303 2/20 0.47
HSD17B10 Q99714 2/20 0.47
MAPT P10636 4/20 0.44
LMNA P02545 2/20 0.44
CRHBP P24387 2/20 0.44
CRHR2 Q13324 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
PDE2A O00408 1/20 0.44
PDE5A O76074 1/20 0.44
ALOX15 P16050 1/20 0.44
NFKB1 P19838 1/20 0.44
APEX1 P27695 1/20 0.44
PDE4A P27815 1/20 0.44
BLM P54132 1/20 0.44
PDE1B Q01064 1/20 0.44
PMP22 Q01453 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27638357 0.85 ALDH1A1 (0.62) ALDH1A1TSHRTDP1CYP3A4ACHE
SCHEMBL1232789 0.83 ALDH1A1 (0.60) ALDH1A1TSHRTDP1CYP3A4ACHE
SCHEMBL9128454 0.83 ALDH1A1 (0.60) ALDH1A1TSHRTDP1CYP3A4ACHE
SCHEMBL5962192 0.82 VCAM1 (0.52) ALDH1A1TSHRTDP1CYP3A4ACHE
SCHEMBL9127741 0.81 ALDH1A1 (0.58) ALDH1A1TSHRTDP1CYP3A4ACHE
SCHEMBL1795352 0.78 TDP1 (0.57) ALDH1A1TSHRTDP1HSD17B10MAPT
SCHEMBL384312 0.77 ALDH1A1 (1.00) ALDH1A1TSHRTDP1CYP3A4ACHE
SCHEMBL29511002 0.77 ALDH1A1 (1.00) ALDH1A1TSHRTDP1CYP3A4ACHE
SCHEMBL5187586 0.77 GPR35 (0.58) ALDH1A1TSHRTDP1HSD17B10MAPT
SCHEMBL5202695 0.77 HSD17B10 (0.62) ALDH1A1TSHRTDP1HSD17B10MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112538053-A Method for synthesizing nitroquinoxaline or derivative thereof and aminoquinoxaline or derivative thereof 同济大学 2021-03-23 CN claimed
CN-110627732-A Method for synthesizing nitroquinoxaline or derivative thereof and aminoquinoxaline or derivative thereof 同济大学 2019-12-31 CN claimed
CN-112538053-B Method for synthesizing nitroquinoxaline or derivative thereof and aminoquinoxaline or derivative thereof 同济大学 2022-09-02 CN disclosed
CN-112538053-A Method for synthesizing nitroquinoxaline or derivative thereof and aminoquinoxaline or derivative thereof 同济大学 2021-03-23 CN disclosed
CN-105753735-B Preparation method of high-efficiency low-toxicity vasopressin antagonist 上海天慈中商药业有限公司 2020-01-17 CN disclosed
CN-110627732-A Method for synthesizing nitroquinoxaline or derivative thereof and aminoquinoxaline or derivative thereof 同济大学 2019-12-31 CN disclosed
CN-105315169-B A kind of preparation method for the treatment of cardiovascular disease drug 上海天慈生物谷生物工程有限公司 2018-12-21 CN disclosed
EP-1720827-A1 METHOD OF PREPARING BENZAZEPINES AND DERIVATIVES THEREOF Centre National de la Recherche Scientifique (FR) 2006-11-15 EP disclosed
WO-2005085183-A1 METHOD OF PREPARING BENZAZEPINES AND DERIVATIVES THEREOF CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2005-09-15 WO disclosed
US-4259350-A PROTECTING DEGRADABLE ORGANIC MATERIAL FROM FUNGAL OR INSECT ATTACK SANKYO COMPANY LIMITED (JP) 1981-03-31 US disclosed