SCHEMBL5717385

SCHEMBL5717385

Fc1cccc(-c2ccccc2)c1Br

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.50
MAPK1 P28482 3/20 0.50
HTT P42858 1/20 0.40
HSD17B10 Q99714 2/20 0.39
HPGD P15428 1/20 0.39
BCL2L1 Q07817 1/20 0.39
CYP2A6 P11509 1/20 0.39
RAB9A P51151 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
MEN1 O00255 1/20 0.39
NPC1 O15118 1/20 0.39
PKM P14618 1/20 0.39
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39
KMT2A Q03164 1/20 0.39
RELA Q04206 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL429933 0.83 ALDH1A1 (0.62) ALDH1A1MAPK1HSD17B10HPGDBCL2L1
SCHEMBL21004874 0.81 L3MBTL1 (0.47) ALDH1A1MAPK1HPGDRAB9ASMN1; SMN2
SCHEMBL31232589 0.80 ALDH1A1 (0.43) ALDH1A1MAPK1HSD17B10HPGDBCL2L1
SCHEMBL201614 0.78 L3MBTL1 (0.50) ALDH1A1MAPK1HTTHSD17B10HPGD
SCHEMBL29356458 0.76 ALDH1A1 (0.68) ALDH1A1MAPK1HSD17B10HPGDBCL2L1
SCHEMBL25644774 0.76 ALDH1A1 (0.54) ALDH1A1MAPK1HSD17B10HPGDBCL2L1
SCHEMBL1627501 0.76 ALDH1A1 (0.68) ALDH1A1MAPK1HSD17B10HPGDBCL2L1
SCHEMBL200742 0.76 ALDH1A1 (0.42) ALDH1A1MAPK1HTTHSD17B10HPGD
SCHEMBL24723508 0.76 ALDH1A1 (0.48) ALDH1A1MAPK1HSD17B10HPGDBCL2L1
SCHEMBL30223212 0.76 CYP1A2 (0.58) ALDH1A1MAPK1HTTCYP2A6RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115703694-A Alkyl substituted fluorene and derivative and preparation method thereof 陕西维世诺新材料有限公司 2023-02-17 CN disclosed
CN-1922156-A Substituted triazoles as sodium channel blockers MERCK & CO INC (US) 2007-02-28 CN disclosed
EP-1689743-A2 PIPERIDINYL-AND PIPERAZINYL-SULFONYLMETHYL HYDROXAMIC ACIDS AND THEIR USE AS PROTEASE INHIBITORS Pharmacia Corporation (US) 2006-08-16 EP disclosed
WO-2005042521-A2 PIPERIDINYL-AND PIPERAZINYL-SULFONYLMETHYL HYDROXAMIC ACIDS AND THEIR USE AS PROTEASE INHIBITORS PHARMACIA CORPORATION (US) 2005-05-12 WO disclosed
EP-1501827-A2 PIPERIDINYL-AND PIPERAZINYL-SULFONYLMETHYL HYDROXAMIC ACID AND THEIR USE AS PROTEASE INHIBITORS Pharmacia Corporation (US) 2005-02-02 EP disclosed
WO-2003091247-A2 PIPERIDINYL-AND PIPERAZINYL-SULFONYLMETHYL HYDROXAMIC ACIDS AND THEIR USE AS PROTEASE INHIBITORS PHARMACIA CORPORATION (US) 2003-11-06 WO disclosed