SCHEMBL5724892

SCHEMBL5724892

Oc1noc2c1C(NCCCC(c1ccccc1)c1ccccc1)CCC2

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.36
HRH1 P35367 1/20 0.36
ALDH1A1 P00352 2/20 0.34
LMNA P02545 2/20 0.34
MAPK1 P28482 1/20 0.34
SOS1 Q07889 1/20 0.34
SCD5 Q86SK9 1/20 0.33
DHODH Q02127 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.32
NPC1 O15118 1/20 0.32
GAA P10253 1/20 0.32
RAB9A P51151 1/20 0.32
EPHX2 P34913 1/20 0.32
KMT2A Q03164 1/20 0.32
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5725148 0.93 SOS1 (0.40) HTR2AHRH1ALDH1A1LMNAMAPK1
SCHEMBL5726290 0.90 SCN5A (0.38) ALDH1A1EPHX2KMT2A
SCHEMBL5725812 0.86 DHODH (0.35) ALDH1A1LMNAMAPK1SCD5DHODH
SCHEMBL5725809 0.86 DHODH (0.35) ALDH1A1LMNAMAPK1SCD5DHODH
Bromide SCHEMBL5725879 0.85 LMNA (0.36) ALDH1A1LMNAMAPK1SCD5DHODH
Bromide SCHEMBL5725876 0.85 LMNA (0.36) ALDH1A1LMNAMAPK1SCD5DHODH
SCHEMBL5724732 0.83 DHODH (0.34) ALDH1A1LMNAMAPK1SCD5DHODH
SCHEMBL5726307 0.83 GRIN2B (0.44) ALDH1A1SMN1; SMN2NPC1GAARAB9A
SCHEMBL5724558 0.83 GRIN2B (0.44) ALDH1A1SMN1; SMN2NPC1GAARAB9A
Bromide SCHEMBL5724922 0.82 GRIN2B (0.43) ALDH1A1SMN1; SMN2NPC1GAARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0812318-B1 4-AMINOTETRAHYDROBENZISOXAZOLE OR -ISOTHIAZOLE COMPOUNDS LUNDBECK & CO AS H (DK) 2006-02-08 EP disclosed
US-6174909-B1 FOR TREATING ANALGESIA, PSYCHOSIS, CONVULSIONS, EPILEPSY, ANXIETY, MUSCULAR AND MOVEMENT DISORDERS, SPASTIC DISORDERS OR SYMPTOMS OF HUNTINGTON'S OR PARKINSONS DISEASE H. LUNDBECK A/S (DK) 2001-01-16 US disclosed
US-5998613-A PSYCHOLOGICAL DISORDERS; ANALGESICS; ANTICONVULSANTS H. LUNDBECK A/S (DK) 1999-12-07 US disclosed